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N-methyl-3-(2-methyl-1H-indol-1-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-(2-methoxyethyl)-3-methyl-4-{[(thiolan-3-yl)carbamoyl]amino}benzamide
(4aS,8aS)-2-[3-(3-hydroxy-3-methylbutyl)benzoyl]-decahydroisoquinolin-4a-ol
methyl N-(4-{5-[(2-methoxyethyl)carbamoyl]furan-2-yl}phenyl)carbamate
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-oxo-N-(pyridin-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-(2-hydroxyethyl)-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-2-one
5-(1H-imidazol-4-ylmethyl)-1,3-diphenyl-1H-1,2,4-triazole
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[2-(4-methylpiperazin-1-yl)ethyl]amine
1-{1-[(2-methylphenyl)methyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
(4aS,8aR)-6-(2-chlorobenzoyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
8-{[2-(trifluoromethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(3-chlorophenyl)cyclopropyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
1-(dimethylamino)-3-[4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]propan-2-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aR,7aS)-N,N-dimethyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-amino-2-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)pyrimidin-4-ol
N-benzyl-1-[1-(2-ethylbutanoyl)piperidin-4-yl]piperidine-3-carboxamide
5-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
methyl 2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetate
N-tert-butyl-1-cyclohexyl-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[(cyclopropylmethyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,2-dihydropyrimidin-2-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
ethyl 1-(cyclohex-3-ene-1-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-(3-hydroxypiperidin-1-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
4-(benzyloxy)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]butanamide
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N3-[2-(4-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R)-N1-(4-cyano-2-ethylphenyl)pyrrolidine-1,2-dicarboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}azepane-2-carboxamide
1-(2-methylpropyl)-5-(3-methylpyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-phenyl-1-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)propan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
6-[({[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)methyl]pyrimidin-4-ol
3-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-4-methoxy-N-methylbenzamide
4-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
2-(4-{[3-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
2-{4-[2-(1H-1,3-benzodiazol-2-ylmethoxy)acetyl]piperazin-1-yl}-N-ethylacetamide
ethyl 1-({[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]carbamoyl}methyl)-1H-imidazole-2-carboxylate
4'-(3,3-dimethylbutyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[2-(1H-indol-4-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4-methylpiperazine
4-ethyl-N,N-dimethyl-6-{4-[3-(pyridin-2-yl)azetidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
methyl[2-(methylamino)ethyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine