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N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(furan-2-ylmethyl)-4-[(2-methoxyethyl)carbamoyl]-1,4-diazepane-6-carboxylic acid
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
(3aS,6aS)-5-{[(furan-2-ylmethyl)carbamoyl]methyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(3-methoxyphenyl)-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{2-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
(3aS,6aS)-1-methyl-N-(thiophen-2-ylmethyl)-octahydropyrrolo[3,4-b]pyrrole-5-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyridin-2-yl)piperidine-4-carboxylic acid
1-[(2,5-dimethylphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
1-(4-methylbenzenesulfonyl)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
ethyl 4-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)benzoate
4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,6-dimethylphenol
2-{3-oxo-9-[3-(pyridin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2,5-dimethyl-1,3-oxazole-4-carboxamide
N-(4-methoxyphenyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(2,3-dimethylphenyl)-N-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
ethyl 6-[3-(2-fluorophenyl)pyrrolidin-1-yl]pyridine-3-carboxylate
2-{N-cycloheptyl-1-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]formamido}acetic acid
2-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methyl-2-(1H-pyrrol-1-yl)propan-1-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3-(cyclohex-1-en-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(3S,7S,8aS)-7-{[(4-chlorophenyl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
[3-(2-methoxyethyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl]methanol
7-(2,3-dimethoxyphenyl)-9-methoxy-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(furan-2-ylmethoxy)phenyl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(4-methoxy-3-methylphenyl)acetamide
(2S)-2-amino-3-(4-hydroxyphenyl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3-benzothiazole-6-carboxamide
4-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]butanoic acid
N-(4-oxo-4H-chromen-6-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
8-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-({2-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}methyl)morpholine
N-methyl-3-(morpholine-4-carbonyl)-N-(oxan-2-ylmethyl)benzene-1-sulfonamide
1-[(2,5-dimethoxyphenyl)methyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
(4aS,7aR)-1-(2,2-dimethylpropyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-butyl-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
2-(1-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
4-(6-methylpyridine-2-carbonyl)-2-(3-phenylpropyl)morpholine
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one