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N-(cyclohexylmethyl)-1-cyclopropyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
7-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-(5-methyl-1,2-oxazol-3-yl)-1-(2-methylpyridin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole-5-carboxamide
5-chloro-2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-fluoropyridine
7-[(2,3-dimethoxyphenyl)methyl]-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[4-(3-benzyl-1H-1,2,4-triazol-5-yl)phenyl]ethane-1-sulfonamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
4-[(diethylamino)methyl]-5-ethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]furan-2-carboxamide
[(3R,4R)-1-[(3-chlorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-ethyl-3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-5-methyl-1H-pyrazole
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)quinoline-3-carboxamide
(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
N-methyl-4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-sulfonyl]thiophene-2-carboxamide
3-(2-cyclopentylethyl)-5-{imidazo[1,2-a]pyridine-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(morpholin-4-yl)-2-oxoethyl]piperidin-3-yl}propanamide
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)urea
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
5-(7-fluoro-2-methylquinoline-4-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
4-{2-[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]ethyl}benzene-1-sulfonamide
(1S,5R)-6-(2-methoxyethyl)-3-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2E)-1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
4-(hydroxymethyl)-N-(2-methoxyphenyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
ethyl 4-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]piperidine
3-(2-amino-4-{[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}-6-methylpyrimidin-5-yl)propanoic acid
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(2-oxopiperidin-1-yl)propanamide
N-[2-(isoquinolin-5-yl)phenyl]-2-methoxyacetamide
1-({1-[6-(3-hydroxypiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
6-[1-(furan-3-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
5,5-dimethyl-3-{2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidine-2,4-dione
(4aR,7aS)-4-(3-cyano-5-fluorobenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}propanamide
N-[3-(cyclohexylsulfanyl)propyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
3-fluoro-6-methyl-N-(4-phenylbutyl)imidazo[1,2-a]pyridine-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-2-[2-(dimethylamino)ethyl]morpholine-4-carboxamide
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
N-{2-[(2-ethyl-6-methylpyrimidin-4-yl)amino]ethyl}pyridine-3-carboxamide
2-methyl-3-(1H-pyrazol-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
1-[7-(furan-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine-3-carbonitrile
N-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(1,3-benzoxazol-2-ylmethyl)(methyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(4-methoxypyrimidin-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-[5-cyclopropyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine