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1-cyclopropyl-4-[4-(2-phenoxyacetyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-{2-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]-4-chlorophenoxy}acetamide
2,3,6-trimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
methyl 4-{[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrazole-3-carboxylate
{4-[(6-methoxynaphthalen-2-yl)methyl]-1-methylpiperazin-2-yl}methanol
2-({4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}methyl)-6,8-dimethylquinolin-4-ol
3-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-ol
1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-{5-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]thiophen-2-yl}acetamide
4-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-N,N-dimethyl-4-oxobutanamide
(4aS,7aR)-1-[(3-chloro-5-ethoxy-4-hydroxyphenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1,3,5-trimethyl-4-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
5-(4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1H-imidazol-2-amine
1-(2-phenoxyethyl)-4-(3,4,5-trifluorophenyl)-1H-1,2,3-triazole
1-cyclopropyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(prop-2-en-1-yl)amino]acetamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N3-cyclooctyl-N5-cyclopropyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4S)-1-(5-cyano-2-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
4-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-ethyl-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-fluoro-2-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amino]methyl}quinolin-4-ol
2-(3-methylbutyl)-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(4-phenyl-1,2,3-thiadiazol-5-yl)piperidine-1-carboxamide
2-(4-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
1-(4-methoxybenzoyl)-4-(4-methyl-1,3-thiazol-2-yl)piperazine
4-ethyl-5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1,3-thiazol-2-amine
4-(2-oxooxolan-3-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
9-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
[3-(1H-imidazol-1-yl)propyl](piperidin-3-ylmethyl)(pyridin-4-ylmethyl)amine
methyl 4-(3-{2-[(4-fluoro-2-methylphenyl)carbamoyl]ethyl}piperidin-1-yl)-4-oxobutanoate
methyl 4-{5-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-1,2,4-oxadiazol-3-yl}benzoate
1-(thiophen-3-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-methylpentyl)morpholine
(2S,4R)-4-amino-N-methyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-2-carboxamide
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-{[methyl(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-3-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
N'-(2-ethoxyphenyl)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]propanediamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]pyridine-2-carboxamide
3-phenyl-8-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,8-diazaspiro[4.5]decan-2-one
(3S,4R)-N,N-dimethyl-4-propyl-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]pyrrolidin-3-amine
5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrazin-2-ol
5-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-N-(propan-2-yl)pyrimidin-2-amine
methyl 5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
7-[(4-ethylpiperazin-1-yl)sulfonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one