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2-(8-methoxy-2H-chromen-3-yl)-1-methyl-1H-1,3-benzodiazole
2-(dimethylamino)-7-[(3-methylthiophen-2-yl)sulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4R)-4-(3-fluorophenyl)-1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
11-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]-7-thia-2,5-diazatricyclo[6.4.0.02,6]dodeca-1(12),5,8,10-tetraene
8-methyl-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(methoxymethyl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)furan-2-carboxamide
1-(3-chlorophenyl)-4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-5-methylpiperazin-2-one
4-benzyl-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N3-ethyl-N5-[(4-methylphenyl)methyl]-N3-(2-methylprop-2-en-1-yl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-6-(5-fluoro-2-methoxybenzoyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-3-(2-fluorophenyl)-N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)prop-2-enamide
1-({4-[1-(dimethylamino)ethyl]phenyl}methyl)-4-phenylpiperidine-4-carbonitrile
2-{3-[(3-chlorophenyl)methyl]-5-[4-(hydroxymethyl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-3-(1-methylpiperidin-3-yl)propan-1-one
2-methyl-5-(2-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)-1,3,4-oxadiazole
(furan-3-ylmethyl)(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
methyl 5-cyano-2-methyl-6-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]pyridine-3-carboxylate
4-hydroxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-5-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-(4-ethylpiperidine-1-carbonyl)-N-(oxan-2-ylmethyl)benzene-1-sulfonamide
3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
7-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl][2-(pyridin-4-yl)ethyl]amine
5-(5-methyl-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]urea
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
8-(3-fluorobenzoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
5-methyl-2-phenyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}furan-3-carboxamide
3-butyl-1-(6-fluoropyridin-3-yl)-3-(furan-2-ylmethyl)urea
5-[3-oxo-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-4-yl]thiophene-2-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
5-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1-(cyclopropylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-5-methyl-1,3-oxazole-4-carboxamide
2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
3-cyclopropyl-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
1-(cyclohexylmethyl)-N5-ethyl-N3-methyl-4-oxo-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
6-(5-chloro-3-fluoropyridin-2-yl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-[2-(dimethylamino)ethyl]-8-[(5-propylfuran-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]propanamide
(1S,5R)-3-(1-methyl-1H-indole-4-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{6-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
N-(3-fluorophenyl)-3-(naphthalene-2-carbonyl)piperidine-1-carboxamide
1-(2-ethylbutyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrrolidine-1-sulfonamide
(5S)-5-{[benzyl({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
4-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}piperazin-2-one
2-(2-fluorophenyl)-2-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}acetic acid
5-acetyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-carboxamide
5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)acetamide