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N-propyl-6-(pyrimidin-5-yl)pyridine-3-carboxamide
5-(azocan-1-yl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-2-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
(2R,6R)-4-(3-chloro-2-fluorobenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{2-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
3-{[(2-ethylbutyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-(cyclopropylmethyl)-1,4-diazepane-6-carboxylic acid
5-methyl-N-[(6-methylpyridin-2-yl)methyl]-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-methoxypyrimidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[(pyridin-3-yl)amino]ethyl}piperidin-2-one
1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
2-(2-{1-[2-(2-chlorophenoxy)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
7-chloro-3-({[(4-fluorophenyl)methyl]amino}methyl)-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
4-[(1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)methyl]morpholine
1-(4-ethylpiperazin-1-yl)-3-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]propan-1-one
9-(2-amino-6-methylpyrimidin-4-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-ethylphenoxy)-1-(4-fluorobenzoyl)azetidine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3,5-dimethyl-1-benzofuran-2-carboxamide
N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]-2,3,6-trimethylquinoline-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
ethyl 5-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
5-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
1-[4-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,3-dihydro-1-benzofuran-7-carboxamide
6-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]-1,4-oxazepan-6-ol
3-(4-methylphenoxymethyl)-1-(1H-pyrrole-2-carbonyl)piperidine
N,N-dimethyl-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]benzene-1-sulfonamide
2-cyclopropyl-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyrimidine
3-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1-[2-(1H-imidazol-1-yl)ethyl]-3-phenylpyrrolidine-2,5-dione
2-{1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}ethan-1-ol
(1R,3S)-7-[6-(hydroxymethyl)pyridine-2-carbonyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-[(6-chloropyridin-3-yl)methyl]-2-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-methylpropanamide
1-cyclopentyl-4-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-2-one
2-methoxy-4-[3-(3-methoxypropyl)piperidine-1-carbonyl]pyridine
N-cyclopentyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
6-ethyl-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-[3-(methylsulfanyl)butyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(2R)-oxolane-2-carbonyl]-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2S,4S)-4-amino-N,N-diethyl-1-[2-(2,3,6-trifluorophenyl)acetyl]pyrrolidine-2-carboxamide
N-(1H-1,2,3-benzotriazol-4-yl)-4-(2-ethylphenyl)piperazine-1-carboxamide
4-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(4aS,7aR)-1-[2-(3-hydroxyphenyl)acetyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
2-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
1-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methoxy-N-(3-{[(1-phenylpiperidin-4-yl)carbamoyl]amino}phenyl)acetamide
[(3-chloro-5-fluoro-4-methoxyphenyl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
4-methoxy-6-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine