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ethyl 1-(1-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-(3-fluorophenyl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
2-[5-(2-chlorophenyl)furan-2-yl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
2-methyl-4-[5-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)thiophen-2-yl]but-3-yn-2-ol
1-(azetidine-3-carbonyl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
(1R,5R)-6-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,4-oxazepan-6-yl)methanol
2-phenyl-7-(1H-pyrazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-tert-butylphenyl)-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N,N-diethyl-1-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(3-methoxypropyl)piperidine-3,5-dicarboxamide
2-(acetamidomethyl)-N-(1H-indol-5-yl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(furan-2-ylmethyl)piperidine-3-carboxamide
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-(2,2,2-trifluoroethyl)piperazine
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}propanoic acid
2-(2-hydroxyethyl)-9-[3-(2-methylphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-ethoxy-2-(1H-imidazol-2-yl)quinoline
2-methoxy-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-(5-chloro-2-fluorobenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
(2S)-1-acetyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]pyrrolidine-2-carboxamide
2-(propan-2-yl)-9-(1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)azetidin-3-ol
methyl 3-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)carbamoyl)amino]-4-methoxybenzoate
2-amino-3-ethyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-(6-chloropyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]quinoline
5-(2-methylphenyl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,2,4-triazin-3-amine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(5-methylpyrazin-2-yl)methyl]amino}acetamide
3-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
(2S)-1-acetyl-N-ethyl-N-(oxan-4-ylmethyl)pyrrolidine-2-carboxamide
4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1,3-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-ethyl-1,6-dimethyl-3-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,4-dihydropyridin-4-one
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
2-{2-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}acetic acid
[1-(4-aminopyrimidin-2-yl)-4-[(4-chlorophenyl)methyl]piperidin-4-yl]methanol
2-amino-6-(4-methyl-1,3-thiazol-5-yl)-4-(1-phenyl-1H-pyrazol-5-yl)pyridine-3-carbonitrile
6-(2H-1,3-benzodioxol-5-yl)-3,4-dihydroquinazolin-4-one
6-phenyl-5-[4-(1H-1,2,3-triazole-5-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N,N-dimethyl-1-(1-methyl-1H-indole-2-carbonyl)azepan-4-amine
3-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1,2-dihydroquinolin-2-one
N-(furan-2-ylmethyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
7-[2-(ethylamino)pyrimidine-5-carbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-3-(morpholin-4-yl)butanamide
{[(3S,4R)-1-(1H-indole-6-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
4-(2-fluoro-5-methoxyphenyl)-6-methylpyrimidin-2-amine
3-ethoxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one