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2-{2-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}-1-(4-methylpiperidin-1-yl)ethan-1-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-indazole-3-carboxamide
{1-[({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
2-(2,4-difluorophenoxy)-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]quinoline
2-tert-butyl-5-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]pyrimidin-4-ol
{5-[2-(2-methoxyphenyl)ethyl]-1-methyl-1H-1,2,4-triazol-3-yl}(phenyl)methanol
5-(3-acetylphenoxymethyl)-N-[2-(propan-2-yloxy)ethyl]-1,2-oxazole-3-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
3-[(dimethylamino)methyl]-1-(2-ethoxybenzoyl)piperidin-3-ol
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)pyridine
1-[(4-chlorophenyl)methyl]-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)benzoic acid
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-methylpropanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-(furan-2-ylmethyl)-N-methylpiperidine-4-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidin-3-ol
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]butanamide
2-{4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-N,N-dimethylacetamide
N-{3-[(2,6-dimethylphenyl)carbamoyl]phenyl}-3-fluoropyridine-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-(furan-2-ylmethyl)piperidine-3-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-(4-{[(dimethylcarbamoyl)(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-3-fluoro-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}benzamide
(3S,4S)-4-({[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)piperidin-3-ol
N-[(5-chlorothiophen-2-yl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-ol
(4S)-N-cyclohexyl-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
(3S,4S)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(1H-imidazol-2-yl)pyrrolidine-3-carboxylic acid
2-(3-fluorophenoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
4-{3-[4-(4-cyanophenyl)-3-oxopiperazin-1-yl]propoxy}benzamide
2-ethyl-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)butanamide
N-methyl-3-(1-methylpiperidin-2-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
4-{5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
N-cyclopropyl-1-(1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
3-(2-methoxyethyl)-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
2-(dimethylamino)-N-[(2-ethoxy-3-methoxyphenyl)methyl]-2-(4-fluorophenyl)-N-methylacetamide
2-[3-methyl-4-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
4-(1H-imidazol-1-yl)-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine-4-carboxylic acid
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
(3S,5R)-1-(3,4-dimethylbenzoyl)-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
(3aS,6aS)-2-(3-methoxypropanoyl)-5-(thiophen-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(morpholine-4-sulfonyl)-5-{pyrazolo[1,5-a]pyridin-7-yl}benzoic acid
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}propanamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(1H-imidazol-2-ylmethyl)-N-methylpropanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol