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(1R,2R,6S,7S)-4-(2,3-dimethoxybenzoyl)-4-azatricyclo[5.2.1.02,6]decane
(2S,4S)-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
8-fluoro-2-{[(1-methanesulfonylpiperidin-4-yl)amino]methyl}quinolin-4-ol
4-[2-(furan-2-yl)pyrimidin-5-yl]-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-{[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]quinoline
2-(2,4-dimethoxyphenyl)-5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-phenylazepane
(2S,4S)-4-amino-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}pyrrolidine-2-carboxylic acid
[(2-methoxy-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl](methyl)amine
3-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}-N-(1,3-thiazol-2-yl)propanamide
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]acetamide
2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(4-cyano-2,5-difluorophenyl)-3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]urea
8-(5-methyl-2-phenylfuran-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-6-methoxy-N-methyl-2,3-dihydro-1H-indene-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
2-[4-(cyclobutylmethyl)piperazin-1-yl]pyridine-3-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)piperidin-2-one
N-(furan-2-ylmethyl)-5-{[2-(4-methoxyphenyl)ethyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(pyridin-3-yl)morpholine
5-[(3-hydroxypiperidin-1-yl)methyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2-oxazole-3-carboxamide
5-methyl-3-(oxan-4-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-{methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}propane-1,2-diol
N-[(3S,4R)-1-[2-(2-ethylphenoxy)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-(2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carbonyl}thiophen-3-yl)acetamide
9-[2-(3-chlorophenyl)-2-hydroxyacetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-(2-phenoxyphenyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
5-fluoro-3-methyl-2-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indole
N-{[4-(dimethyl-1,2-oxazol-4-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N4-ethyl-N2-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
4-(4-methoxyphenoxy)-1-(thiophen-3-ylmethyl)piperidine
5-(methoxymethyl)-N-(4-{5-methyl-4-[(2-methylpropanamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-2-carboxamide
N3-(cyclopropylmethyl)-N5-ethyl-1-(2-methylpropyl)-4-oxo-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
(1R,5R)-6-(3-chlorothiophene-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N,N-dimethyl-2-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-2,3-dihydro-1H-inden-2-amine
2-fluoro-N-{[(2S,4S)-4-fluoro-1-[(2S)-2-(methylamino)propanoyl]pyrrolidin-2-yl]methyl}benzamide
1-{1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}-3-methylbutan-1-ol
3-[2-(4-fluorophenyl)ethyl]-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
4-[(2-methylpiperazin-1-yl)methyl]-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)benzamide
2-benzyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzoxazole-5-carboxamide
2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}propanamide
5-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
2-[2-(dimethylamino)-2-(4-methylphenyl)acetamido]-2-methylpropanamide
1-(2-{3-[(2-methoxyphenyl)methyl]-1-propyl-1H-1,2,4-triazol-5-yl}ethyl)-1H-1,2,3,4-tetrazole
5-(4-fluorophenyl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,2,4-triazin-3-amine