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2-phenoxy-N-[4-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
2-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
(1R,5R)-3-(4-chlorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amine
1-[(5-chlorothiophen-2-yl)methyl]-8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decane
1-{[4-(cyclopentyloxy)phenyl]methyl}-3-(methoxymethyl)pyrrolidine
1-butyl-5-[1-(3-methoxyphenoxy)ethyl]-3-methyl-1H-1,2,4-triazole
1-[2-(1H-imidazol-1-yl)ethyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoacetamide
[(2-fluoro-4-methoxyphenyl)methyl]({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amine
N-(2-fluoro-4-methylphenyl)-2-[2-(furan-2-yl)-2-oxoacetamido]propanamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)propan-1-one
5-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylic acid
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
N-[(3S,4R)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-({1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxopropan-2-yl}sulfanyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetamide
1-(2-methoxyethyl)-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
2-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1H-indole-3-carboxamide
2-(2,4-dichlorophenoxy)-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]acetamide
1-[(3-methoxyphenyl)methyl]-4-[2-(methylamino)pyridine-3-carbonyl]piperazin-2-one
2-(methylamino)-1-[4-(4-methylphenoxy)piperidin-1-yl]ethan-1-one
4-chloro-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)thian-4-amine
[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)sulfamoyl](ethyl)methylamine
(3R,4R)-4-amino-1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-3-ol
1-(2,4-difluorobenzoyl)-4-(3-phenylpropyl)-1,4-diazepane
N-[(2-chlorophenyl)methyl]-N-ethyl-3-[(2-fluorophenyl)formamido]propanamide
2-{2-[(5-oxo-1-propylpyrrolidin-3-yl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-[(1-methyl-1H-indol-6-yl)methyl]-8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decane
ethyl 1-(pyridin-4-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
methyl (2S,4R)-4-(4-methylbenzamido)-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetamide
2-(3-methoxypropyl)-9-(3-methylbenzenesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
1-(2,4-difluorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
N-cyclopentyl-1-methyl-5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,6-dimethyl-2-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrimidin-4-amine
2-[2-(azepan-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{6-hydroxy-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4-diazepan-1-yl}-2-phenylethan-1-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(3-ethoxypropyl)-3-methoxybenzamide
2-(3-methoxyphenyl)-2-{methyl[(5-methylfuran-2-yl)methyl]amino}acetic acid
[3-(hydroxymethyl)-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-3-yl]methanol
6-benzyl-1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octane
N-[3-(1H-imidazol-1-yl)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine