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6-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyridine-3-carbonitrile
N-(2,3-dihydro-1H-inden-2-yl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-(2-hydroxypropyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(3-methylbenzoyl)piperidine-3-carboxylate
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
4-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzoic acid
3-[5-(dimethylamino)-1H-1,2,4-triazol-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-(oxolan-2-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
2-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]acetic acid
5-{3-[(2-methoxyphenyl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-N-methylpyrimidin-2-amine
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N1,N1-dimethyl-N3-{3-[(pyridin-3-yl)amino]propyl}piperidine-1,3-dicarboxamide
9-methyl-3-{7-methylthieno[3,2-d]pyrimidin-4-yl}-3,9-diazaspiro[5.6]dodecan-10-one
4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-2-ethylmorpholine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-methylpyridine-3-carbonyl)piperidin-3-yl]propan-1-ol
2-[(4aR,7aS)-4-(4-methyl-1H-imidazole-2-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-{4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazin-1-yl}pyrimidine
4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1-(2-methylphenyl)piperazin-2-one
N-{4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}acetamide
1-[3-(1H-imidazol-1-yl)propyl]-2-(4-methoxynaphthalen-1-yl)-1H-imidazole
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-2-phenylpiperazine
1-{1-[(2-fluoro-5-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[3-(3-fluorophenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(methylsulfanyl)benzamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-2,1,3-benzoxadiazole-5-carboxamide
3-(1-benzylazetidin-2-yl)-4-(3-methylphenyl)-4H-1,2,4-triazole
(1S,6R)-3-methyl-9-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,4S)-4-cyclopropyl-1-[1-(4-fluorophenyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}but-3-en-1-one
(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]sulfonyl}phenyl)urea
2-(5-hydroxypyrazine-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
2-[(4-methyl-1,3-thiazol-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[1-(1-benzoxepine-4-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
4-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}pyrimidine
4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1-propyl-1H-pyrazole
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-[2-(pyrazin-2-yl)ethyl]urea
1-(azepan-1-yl)-3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropan-1-one
7-(2-hydroxy-5-methylbenzoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4S)-N-ethyl-4-[2-(2-ethyl-1H-imidazol-1-yl)acetamido]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
1-cyclopropanecarbonyl-4-(pyrazin-2-yl)-1,4-diazepane-6-carboxylic acid
2-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
{4-methyl-5-[(1-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperidin-4-yl)methyl]-4H-1,2,4-triazol-3-yl}methanol
N-[1-(4-chlorophenyl)cyclobutyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(4-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
N-cyclopropyl-3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
3-[(cyclobutylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one