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N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-7-fluoro-2-methylquinoline-4-carboxamide
(3S,9aR)-8-(3-methylbutyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(2E)-N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(oxolan-2-ylmethyl)pyrazine-2-carboxamide
4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-1-phenylpiperazin-2-one
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
N-(3-chloro-4-fluorophenyl)-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]propanamide
3-methyl-4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethoxy]-1,2,5-oxadiazole
N-cyclopropyl-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
1-(2-fluorophenyl)-4-[4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]piperidin-4-ol
5-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)-1-azabicyclo[3.2.1]octane
2-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-cyclopropylpyridine-4-carboxamide
methyl 5-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-(4-chlorophenoxy)-N-(pentan-3-yl)piperidine-4-carboxamide
diethyl({3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
5-[(3,5-dimethoxyphenyl)methyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
1-cyclopentyl-4-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperazin-2-one
3-{[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)sulfamoyl}-N-methyl-N-propylbenzamide
2-(4-fluorophenyl)-2-hydroxy-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-(2-{3-[3-(2-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine
2-(1H-indol-3-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
9-(4-methylpyridine-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazin-2-ol
methyl 2-[3-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-1H-indol-1-yl]acetate
1-(3,4-dimethylphenyl)-5-(1,4-dioxan-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
(2S)-2-amino-3-hydroxy-1-[4-(thiomorpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
3-(2-amino-5-methylpyrimidin-4-yl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
3-methyl-9-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-3,9-diazaspiro[5.6]dodecane
4-[(4-chlorophenyl)methyl]-3-[(4-methylpiperazin-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N,1-tris(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-9-[5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-methylazepane-2-carboxamide
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-ol
[(2-chloro-4,6-dimethoxyphenyl)methyl][(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
(3R,4S)-4-(4-methoxyphenyl)-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-amine
1-(4-{[3-(diethylamino)propyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(2S)-N-methyl-2-(methylamino)-N-[(4-phenoxyphenyl)methyl]propanamide
[3-(cyclopropylmethyl)-1-(5-ethylthiophene-3-carbonyl)piperidin-3-yl]methanol
N-cyclohexyl-3-fluoro-7-methyl-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(1H-1,3-benzodiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(6-methoxypyridin-2-yl)-2-{[(2-phenylethyl)amino]methyl}phenol
5-{3-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-5-methylpyrrolidin-2-one
benzyl 4-[(3-hydroxypiperidin-3-yl)methyl]-1,4-diazepane-1-carboxylate
N-benzyl-2-(4-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
7-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one