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1-(2-{[(5-acetamido-2-methoxyphenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
N3-methyl-1-(3-methylbutyl)-4-oxo-N5-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-{3-[2-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-3-oxopropyl}acetamide
2-(2,5-dimethylphenyl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
(3S,4S)-1-(2,6-dimethylquinoline-3-carbonyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
(2R,6R)-4-(morpholine-4-sulfonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
[(1-ethyl-1H-pyrazol-4-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(propan-2-yl)amine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-(3,4-dimethylphenyl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-amine
2-{2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-1H-imidazole
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(morpholin-3-yl)acetamide
4-benzyl-1-(2-ethoxyethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidine
methyl 7-oxo-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1,3-dihydroxypropan-2-yl)-2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
2-(1H-1,2,3,4-tetrazol-5-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-[3-(morpholin-4-yl)propyl]acetamide
3-[2-(3-methoxyphenyl)ethyl]-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
5-{4-hydroxy-1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
2-({5-fluoro-2-[3-(methylsulfanyl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
1-(4-methoxyphenyl)-2,2-dimethyl-N-[3-(3-oxopiperazin-1-yl)propyl]cyclopropane-1-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2,2-diphenylethyl)-4-(4-methyl-1H-pyrrole-2-carbonyl)morpholine
1-[1'-(5-chloropyridin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
4-chloro-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
7-[2-hydroxy-4-(methylsulfanyl)butanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-methyl-5-propyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
6-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-2,3-dihydropyridazin-3-one
5-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-3-(1H-pyrazol-1-yl)benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
{1-[2-(2-aminoethyl)quinazolin-4-yl]-3-ethylpiperidin-3-yl}methanol
4-(furan-2-ylmethyl)-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-ethyl-1-methyl-3-[1-(1,8-naphthyridine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (2S)-1-(3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)pyrrolidine-2-carboxylate
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-ethoxy-5-(2-{[(1s,4s)-4-aminocyclohexyl]amino}pyrimidin-4-yl)benzoic acid
2-chloro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
2-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
(1S,5R)-3-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,4-dimethyl-N-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-{3-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
methyl 1-[(3S,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-(propan-2-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-{[4-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinolin-8-ol
(1R,5S)-6-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-6-azabicyclo[3.2.1]octane
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-4-ol
5-tert-butyl-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,3-benzodiazole