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3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
N-cyclopentyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(2E)-N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(pyridin-2-yl)-N-(pyridin-3-ylmethyl)prop-2-enamide
3-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[2-(methylsulfanyl)phenyl]urea
N-(4-methoxyphenyl)-1-(quinoxalin-2-yl)piperidin-3-amine
2-[(3-chlorophenyl)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
3-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]aniline
N,N-dimethyl-2-[(1S,5R)-3-(6-methyl-2-propylpyrimidin-4-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-{1H-imidazo[4,5-c]pyridin-2-yl}-3-(3-methoxyphenyl)-1-phenyl-1H-pyrazole
1-(2-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}ethyl)imidazolidin-2-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-[4-({[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
N-[2-(1,3-thiazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3,5-dimethoxybenzamide
1-(4-chlorophenyl)-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}cyclopropane-1-carboxamide
N-ethyl-7-methoxy-N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
3-ethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,2-oxazole-5-carboxamide
7-chloro-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
5-(6,6-dimethyl-5-oxothiomorpholine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
1-[3-({[7-chloro-2-(2,3-dimethoxyphenyl)quinolin-3-yl]methyl}amino)propyl]pyrrolidin-2-one
6-{[(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amino]methyl}-1,4-oxazepan-6-ol
2-{2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-6-methylpyridine-3-carbonitrile
[2-(3,5-difluorophenyl)ethyl](methyl)[2-(morpholin-4-yl)propyl]amine
4-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
3,5-difluoro-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]pyridine-2-carboxamide
8-[(2-butyl-1H-imidazol-4-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
5-[2-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]imidazolidine-2,4-dione
3-(2,5-dimethoxyphenyl)-1-[2-(methylsulfanyl)benzoyl]pyrrolidine
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-{[1-(4-methoxyphenyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2,3-dimethyl-6-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}quinoxaline
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)but-2-ynamide
4-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
3-(1-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}piperidin-4-yl)-N-(3-methylphenyl)propanamide
(3R,4R)-4-(azepan-1-yl)-1-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-3-ol
(3R,4R)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-benzyl-N3-[(4-methoxyphenyl)methyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[methyl(1,2-oxazol-3-ylmethyl)amino]-2-[3-(methylsulfanyl)phenyl]acetic acid
1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(3-fluorophenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-(5-{[3,5-dichloro-4-(propan-2-yloxy)phenyl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-methyl-4-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyridin-2-amine
2-{[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide