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N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-fluoro-6-methoxybenzamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]oxolane-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(4-methylnaphthalen-1-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(1S,5R)-3-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
5-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-methyl-6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
3-[(2-fluorophenyl)formamido]-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylpropanamide
5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]pentanoic acid
3-{3-methyl-5-[4-methyl-2-(pyridin-3-yl)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-(cyclohexylmethyl)-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-benzoyl-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
3-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-1,2-benzothiazole
4-[3-(2-butoxy-5-methylphenyl)-1-methyl-1H-1,2,4-triazol-5-yl]morpholine
1-[(5-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}furan-2-yl)methyl]-1H-imidazole
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[2-(morpholin-4-yl)ethyl]-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidin-2-one
(1R,5R)-6-(cyclopropylmethyl)-3-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane
4-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(5-tert-butyl-1H-pyrazol-3-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(pyrazin-2-yl)acetamide
3-(1,3-benzothiazol-2-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{1,4-dioxa-8-azaspiro[4.5]decan-8-yl}-4-[2-(4-fluorophenyl)pyrrolidin-1-yl]butane-1,4-dione
2-cyclopropyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]propan-1-one
1-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-2,3-dihydro-1H-indole
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-methyl-1-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]urea
1-{[1-(pyrazine-2-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
6-(difluoromethyl)-2-[3-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyrimidin-2-ylmethyl)amine
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(1H-imidazol-1-yl)acetamide
7-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}cyclobutan-1-amine
2-{1-[(4-fluorophenyl)methyl]-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-(5-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
1-[(4aR,8aS)-1-[4-(piperidin-1-yl)benzoyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
(1S,2R)-1-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-2,3-dihydro-1H-inden-2-ol
4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
2-[5-(5-chlorothiophen-2-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
9-methoxy-N-methyl-3-{9-methyl-9-azabicyclo[3.3.1]nonan-3-yl}-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
5-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
1-(adamantan-1-yl)-4-(3-methyl-1,2-oxazole-5-carbonyl)piperazine
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
2-methanesulfonamido-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide