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2-amino-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide
1-(1-benzofuran-5-ylmethyl)-4-[(3-methylphenyl)methyl]piperazine
2-[1-(pyrrolidin-1-yl)cyclohexanecarbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1,2-dihydroquinoxalin-2-one
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-phenyl-3-(piperidin-4-yl)-1-(pyrimidin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
6-chloro-2-(3,5-dichloropyridin-4-yl)-1H-1,3-benzodiazole
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(1H-imidazol-2-ylmethyl)amino]methyl}piperidin-2-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(3-cyclopentylpropyl)propanamide
9-[(3,4-difluorophenyl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(2,6-dihydroxybenzamido)-N-phenylpiperidine-1-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[4-(dimethyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
1,4-dimethyl-9-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-1,4,9-triazaspiro[5.5]undecane
N-methyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}pyrrolidine-3-carboxamide
2-{[(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)oxy]methyl}pyridine
N3-[(5-chlorothiophen-2-yl)methyl]-1-cyclohexyl-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-hydroxy-1-methyl-3-({[3-(methylsulfanyl)propyl]amino}methyl)piperidin-2-one
N-[3-(cyclohexyloxy)propyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(thiophene-2-carbonyl)piperidine
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
(4aS,8aR)-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
[1-(2-fluoro-5-methylbenzoyl)piperidin-4-yl](pyridin-2-yl)methanol
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(2-methoxyethyl)-1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
4-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]-N-methylbenzene-1-sulfonamide
8-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-ethyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(1-methyl-1H-pyrazole-5-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(3-methoxy-2-propoxyphenyl)methyl]pyrimidin-2-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
5-(3,5-dimethyl-1H-pyrazol-4-yl)-3-(4-methoxyphenyl)-1,2,4-oxadiazole
1-(4-methoxyphenyl)-3-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-2-one
3-{[(2,4-dichloro-3-methylphenyl)carbamoyl](methyl)amino}-N-methylbutanamide
4-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
(4S)-4-(propan-2-yl)-3-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazolidin-2-one
3-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)-1,2-benzothiazole
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-[(3,4-difluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-5-{1-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-amine
N,2-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzothiazole-6-carboxamide
2-{2-[(2-methoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
(3S,4S)-1-{3-[4-(dimethylamino)phenyl]propanoyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid