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(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
butyl 3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxylate
1-(3-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
4-[4-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
N-cyclopentyl-N-{[3-methoxy-4-(oxan-2-ylmethoxy)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)benzamide
1-{2-hydroxy-3-[4-methoxy-2-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
(3R,4R)-3-cyclobutyl-4-methyl-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-ol
(1,4-dioxan-2-ylmethyl)(methyl)[(2,5,7-trimethylquinolin-4-yl)methyl]amine
1-[1-(5-chloro-3-fluoropyridin-2-yl)piperidin-4-yl]piperidin-4-ol
N-(pyridin-2-ylmethyl)-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazine-2-carboxamide
methyl 1-(2-methoxyethyl)-5-{[1-(methylsulfanyl)propan-2-yl]amino}-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
2-amino-6-{4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
3-(4-ethylphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1H-pyrazole-5-carboxamide
1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
N-methyl-5-propyl-N-(quinolin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-hydroxyazepan-4-yl]methyl}methanesulfonamide
(1R,5S)-6-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-chloro-4-hydroxyphenyl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
2-(2-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)-1,3-thiazole
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(4-fluorophenyl)-2-hydroxyethan-1-one
dimethyl({[6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-3-yl]methyl})amine
N-[1-(2,2-diphenylethyl)piperidin-4-yl]methanesulfonamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methylpropyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(furan-2-ylmethyl)acetamide
2-[1-({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}methyl)piperidin-3-yl]propan-2-ol
3-methyl-5-(2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(5-fluoro-2-methylphenyl)acetamide
N-cycloheptyl-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,5R)-6-(4-methoxy-2-methylbenzoyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(3-methoxyphenyl)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)morpholine
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-ethyl-6-(1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-hydroxy-5-methylbenzamide
(4aR,7aS)-1-(2,2-dimethylpropanoyl)-4-(6-methylpyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-3-propylmorpholine-4-sulfonamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(morpholin-4-yl)ethyl]butanamide
5-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-2-one
1-(dimethylamino)-2-(4-{[4-(propan-2-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
6,6-dimethyl-1-(2-methylphenyl)-N-[1-(propan-2-yl)piperidin-4-yl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
ethyl 4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
2-(2-{1-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
1-(3-fluorophenyl)-6,6-dimethyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1,7-dimethyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole-2-carboxamide