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7-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1,3-diazepane-2,4-dione
2-(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)-5-methylpyrazine
(3S,4R)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-(2-chloro-6-methylphenyl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
5-[3-(benzyloxy)piperidine-1-carbonyl]thiophene-2-carboxylic acid
3-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
4-[2-(4-chlorophenoxy)acetyl]-1-(2-methylphenyl)piperazin-2-one
9-[2-(3-fluorophenyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[5-(1-methanesulfonylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-(pyridine-4-carbonyl)piperidin-4-amine
ethyl 3-[(3-methoxyphenyl)methyl]-1-(2-oxo-2-phenylacetyl)piperidine-3-carboxylate
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-methyl-N-[2-(3-methylthiophen-2-yl)ethyl]-2-(thiophen-2-ylformamido)propanamide
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(2-methoxyphenyl)methyl]piperazine
4-(4-fluoro-2-methylphenoxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
5-ethyl-2-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}pyridine
2-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-[1-(4-methanesulfonylphenyl)cyclobutyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,3,5-trimethylfuran-2-carboxamide
(2R,3R)-3-[4-(4-fluorophenyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1-methyl-6-oxopiperidin-3-yl)benzamide
3-(2-methylphenyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
2-(4-fluorophenoxy)-1-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
4-chloro-N-[2-(4-ethylmorpholin-2-yl)ethyl]-3-fluorobenzamide
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-2-yl)acetamide
2-(2,3-difluorophenyl)-1-(1-methoxybutan-2-yl)-1H-imidazole
(3S,4R)-1-acetyl-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
1-(2-chloro-5-sulfamoylphenyl)-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
ethyl 4-(2-phenoxyethyl)-1-(1-phenylpiperidin-4-yl)piperidine-4-carboxylate
N-[(4-hydroxyphenyl)methyl]-2-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
9-(3-acetylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-2-(oxolan-2-yl)-1H-1,3-benzodiazole
N-cyclopentyl-6-(8-methoxyquinolin-5-yl)pyridazin-3-amine
2-methylpropyl N-[(3R,5S)-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-3-yl]carbamate
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-1-(4-phenylpiperidin-1-yl)ethan-1-one
N-(4-{2-oxo-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethyl}phenyl)cyclopropanecarboxamide
1-{3-[3-(hydroxymethyl)-8-methylquinolin-2-yl]phenyl}ethan-1-one
5-methoxy-1-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-indole-2-carboxamide
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(furan-2-yl)-N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-oxoacetamide
3-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{4-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]piperidin-1-yl}pyridine-3-carbonitrile
(3S,4R)-1-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-3-ethyl-4-methylpiperidin-4-ol
5-tert-butyl-N-{2-[methyl(phenyl)amino]propyl}-1,3,4-oxadiazol-2-amine
(2S)-3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propane-1,2-diol
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-(pyrazin-2-yl)propanamide
1-[3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]ethan-1-one