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N-[2-(4-chlorophenoxy)ethyl]-N-(furan-2-ylmethyl)-2-(2-oxoimidazolidin-1-yl)acetamide
ethyl 5-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}furan-2-carboxylate
1-[2-({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-methoxy-4-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]pyridine
methyl (1R,3S,3aR,6aS)-3-(3-ethenylphenyl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
(2S,4R)-4-(4-{[1-(2,3-dimethylphenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-ethylpyrrolidine-2-carboxamide
5-cyclopropanecarbonyl-1'-[(2-fluoro-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(methylamino)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyridine-4-carboxamide
methyl 6-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-3-(1-phenylcyclopropaneamido)thieno[2,3-b]pyridine-2-carboxylate
N-(2-hydroxyethyl)-3-(1-methylpiperidin-2-yl)-N-(thiophen-2-ylmethyl)propanamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-benzyl-N-ethyl-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
1-(2-hydroxyethyl)-4-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-1,4-diazepan-6-ol
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}quinoxaline
1-(1-benzofuran-2-ylmethyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
4-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-1-methylpiperazin-2-one
4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]butanamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
1-(4-{1-[(2,4,6-trifluorophenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)butan-2-ol
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[1-(furan-2-yl)ethyl]acetamide
(3aS,6aS)-2-acetyl-5-{[4-(2-methylpropyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(4-fluoro-2-methoxyphenyl)-1H-1,3-benzodiazole
N-{[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2-{4-[(8-methoxy-2H-chromen-3-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-(3-phenylpropyl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
4-[4-(3-fluorophenoxy)piperidine-1-carbonyl]pyridine
1-cyclohexyl-6-hydroxy-4-[(1-methyl-1H-indol-3-yl)methyl]-1,4-diazepan-2-one
3-[1-(piperidin-3-yl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-4-methylpyrimidine-5-carboxamide
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyridin-4-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-hydroxy-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
(3aR,7aS)-2-(7-methyl-1-benzofuran-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)acetamide
(3S,4R)-1-(3-chloro-4-methoxybenzoyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}propanamide
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-fluorophenyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}azetidine
2-(methylamino)-N-{1-[(4-methylphenyl)methyl]cyclopropyl}pyrimidine-5-carboxamide
methyl (2S,4R)-4-hydroxy-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidine-2-carboxylate
N-[(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
7-methoxy-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1,2,3,4-tetrahydronaphthalen-2-amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2-fluoro-5-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(benzylsulfamoyl)[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]amine
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidine
(3R,4R)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}({1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
9-hydroxy-2-{[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N2-(2-methoxyethyl)-N4-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine