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(4aR,7aS)-4-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-(2-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(thiophene-2-carbonyl)-1,4-diazepan-6-yl]oxy}acetamide
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-methoxyethyl)piperazine
1-(2-hydroxypyridin-3-yl)-3-(2-methoxyethyl)-3-(1,3-thiazol-2-ylmethyl)urea
3-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)quinoline
2-phenyl-1-{1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl}ethan-1-one
1-[3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]piperidin-3-ol
3-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,3-oxazolidin-2-one
(5S,9aS,9bS)-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[(3S,5R)-1-(2-methyl-1H-pyrrole-3-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2,2-dimethyl-3-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-1-ol
3-(3-chlorophenyl)-1-(4-hydroxypiperidin-1-yl)-3-phenylpropan-1-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
[(6-fluoroquinolin-2-yl)methyl][2-(1H-imidazol-1-yl)ethyl]methylamine
1-(2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
2-cyclopentyl-N-[2-(3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxy)propyl]acetamide
1-phenyl-4-(1-propylpiperidin-4-yl)-1,4-diazepane
3-(azocan-1-yl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-(1-methyl-6-oxopiperidin-3-yl)-4-(piperidin-1-ylmethyl)benzamide
ethyl 1-[(6-methoxy-2H-chromen-3-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
2-methyl-6-[1-(quinolin-4-ylmethyl)piperidin-3-yl]pyrimidin-4-ol
3-(3-{[(2-hydroxy-3-phenylpropyl)amino]methyl}-1H-indol-1-yl)propanamide
(2R,3R)-3-amino-1'-(3-methyl-1H-indole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(2-methyl-1-{4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}propan-2-yl)morpholine
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}oxolane-3-carboxamide
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(2-phenylethyl)acetamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
2-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(4-methoxyphenyl)ethyl]-N-methylbenzamide
1-[4-(methylsulfanyl)butan-2-yl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-6-(4-methoxyphenyl)-1,2-dihydropyridin-2-one
2-amino-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-[(2-fluorophenyl)formamido]propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
2-(2,3-difluorophenoxymethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-oxazole
1,3-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
2-{[3-(4-chlorophenoxy)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(3S,9aR)-3-benzyl-8-[(2-fluoro-5-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-[(4-phenoxyphenyl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
7-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-4-methyl-2H-chromen-2-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3,5-dimethoxy-N-(pyridin-4-ylmethyl)benzamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(methanesulfonylmethyl)piperidine
(4aS,8aS)-2-(5-methyl-1,2-oxazole-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(4-ethenylbenzoyl)-2-[(4-fluorophenyl)methyl]morpholine