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1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-methyl-N-(pyridin-2-ylmethyl)pyridin-2-amine
2-[5-(2H-1,3-benzodioxol-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-6-methylpyridine
[4-(oxan-2-ylmethyl)-1-(quinoxalin-5-ylmethyl)piperidin-4-yl]methanol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,2,6-trimethylquinoline-4-carboxamide
methyl 2-[N-methyl-1-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]acetate
(1R,5R)-3-methanesulfonyl-6-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H-pyrrole-2-carboxamide
(1R,5R)-N,N-dimethyl-6-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,3-benzodiazole
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
(5S)-5-{3-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-({1-[(2-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1,4-diazepan-5-one
4-chloro-N-[1-(2-methoxyphenyl)ethyl]-N,1-dimethyl-1H-indole-2-carboxamide
1-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
5-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
9-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-benzyl-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-[(1-methylpiperidin-4-yl)oxy]-N-propylaniline
1-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-(3-methylbutyl)-N3-(2-methylpropyl)-N5-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,2R,6S,7S)-4-(5-propyl-1,2,4-oxadiazol-3-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-cyclopentyl-N,N-diethyl-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
N-(quinolin-3-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(4-methoxybenzoyl)piperazine
1-(2-methoxyethyl)-3-methyl-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-(2-oxopyrrolidin-1-yl)benzamide
3-propyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
8-(2-cyclopropylpyrimidine-5-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-[1-(1-methylpiperidin-4-yl)piperidine-3-carbonyl]azepane
methyl (2S,4S,5R)-4-[(2-acetamidoethyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
[(2,5-difluorophenyl)methyl]({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)pyridine
1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(1-methyl-1H-indazol-5-yl)urea
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
ethyl 1-(1H-1,3-benzodiazole-5-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-1H-imidazole-2-carboxamide
(3aR,6aS)-2-methyl-5-[(5-phenylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole
3,4,7-trimethyl-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
3-[2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
3-[4-(2-methoxyphenyl)phenyl]-1-(morpholin-2-ylmethyl)urea
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(1-methyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]morpholin-2-yl}ethyl)cyclohexanecarboxamide