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{2-[2-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
2-(2,6-difluorophenyl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
1-[2-(3-fluorophenyl)ethyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
1-[(5-methylfuran-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1,3-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-({1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
4-(2,8-dimethylquinoline-4-carbonyl)-1,4-oxazepan-6-ol
(2S)-2-amino-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
1-[2-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(3R,4R)-4-(azepan-1-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-ol
(3S,4R)-1-{[3-(difluoromethoxy)phenyl]methyl}-4-methylpiperidine-3,4-diol
1-{1-[2-(methylcarbamoyl)ethyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
methyl 1-({4-[(2-methoxyethyl)amino]-8-methylquinazolin-2-yl}methyl)piperidine-2-carboxylate
2-{4-[(3-methoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(1S,5R)-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[2-(1H-imidazol-4-yl)ethyl]-9-(morpholine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
8-[5-(dimethyl-1,2-oxazol-4-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]quinoline
(5-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
5-[(4-fluorophenyl)methyl]-5-{3-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-benzyl-N-(oxolan-2-ylmethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(2S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-methyl-4-[(pyrimidin-2-yl)amino]pyrrolidine-2-carboxamide
3-[2-(2-hydroxyethoxy)ethyl]-1-(2-methyl-1-benzofuran-5-yl)urea
2-[2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethoxy]ethan-1-ol
3-chloro-5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyridine
N-[3-(furan-2-yl)phenyl]-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxamide
1-{2-[2-(4-chlorophenyl)morpholin-4-yl]pyrimidin-4-yl}piperidin-4-ol
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-methyl-2-oxopentanamide
methyl 1-methoxy-2-oxo-8-[2-(phenylsulfanyl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
(1S,5R)-3-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(cyclopropylmethyl)-2-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-[(dimethylamino)methyl]-1-(5-fluoro-2-methylbenzoyl)azepan-4-ol
2-(3-{[methyl(3,3,3-trifluoropropyl)amino]methyl}piperidin-1-yl)ethan-1-ol
6-(2,6-dimethoxyphenyl)-N-ethylpyridine-3-carboxamide
9-[2-(methylsulfanyl)propanoyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-5-methylpyrazine
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N,N-dimethylacetamide
{1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methanol
methyl 5-methyl-4-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxylate
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N,1-dimethyl-N-(1,2-oxazol-5-ylmethyl)-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-2-methyl-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(1-benzylpiperidin-4-yl)methyl]-N,1-dimethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(piperazin-1-yl)ethan-1-one
N-[2-(ethanesulfonyl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-(4-{[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl}phenyl)acetamide