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N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl]pyridine-3-carboxamide
3-(2-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazolidin-2-one
6-cyclopentyl-N-(1H-indol-4-ylmethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(quinoxalin-6-ylmethyl)propanamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-4-(1H-1,2,4-triazol-3-yl)benzamide
1-{5-[3-(1H-pyrazol-3-yl)phenyl]furan-2-carbonyl}piperidine
4-(2-methoxyphenoxy)-1-[4-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
4-(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)piperazin-2-one
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
8-(5-methyl-4-phenylthiophene-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl 4-{[2-(2-aminoethyl)quinazolin-4-yl]amino}butanoate
2-(2-methyl-1H-indol-3-yl)-1-(4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)ethan-1-one
1-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}piperidin-3-ol
methyl 1-[(3S,5S)-5-[(furan-2-ylmethyl)carbamoyl]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-{2-[2-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[4-(2,4-difluorophenyl)-5-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N-methylpyrimidin-4-amine
2-({4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}methyl)benzonitrile
(2R,4S)-4-hydroxy-1-[3-(2-methoxyphenyl)benzoyl]piperidine-2-carboxylic acid
N-[(3S)-1-benzylpiperidin-3-yl]-2-(ethylamino)pyrimidine-5-carboxamide
1-(piperidin-1-yl)-2-{3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-one
3,5-dimethoxy-N-({1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)benzamide
3-{[(5-methyl-1,2-oxazol-3-yl)formamido]methyl}-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(thiophen-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-(carbamoylmethyl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide
5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyridine-2-carbonitrile
4-[2-ethyl-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
3-(1H-indol-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
3-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1-propyl-1H-pyrazole
2-[(4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)methyl]pyridine
N-[(1-benzylpiperidin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-ethyl-4-{[(1-propylpiperidin-4-yl)amino]methyl}hexanenitrile
2-chloro-N-{2-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
(2S,3R)-2-amino-3-hydroxy-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
3-(cyclopropylmethyl)-1-[2-(pyridin-3-yl)acetyl]piperidine-3-carboxylic acid
2-[2-(trifluoromethyl)morpholin-4-yl]-1,3-benzothiazole
1-{2-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-ethyl-5-{4-phenyl-1-[2-(piperidin-1-yl)ethyl]-1H-imidazol-5-yl}pyrimidine
3-(2,4-difluorophenyl)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(pyridin-4-yl)propanamide
2-methyl-4-(3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one
1-(5-ethoxyfuran-2-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one