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2-methyl-1-{3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
2-(4-fluorophenyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-cyclopropyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
1-[(5-chlorothiophen-2-yl)sulfonyl]-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
1-methyl-2-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(3S,4S)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
propan-2-yl 5-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanamido]-2-chlorobenzoate
2-{3,5-dimethyl-4-[2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoacetamido]-1H-pyrazol-1-yl}acetic acid
5-{[2-(naphthalen-2-yloxy)propanamido]methyl}thiophene-2-carboxylic acid
1-(4-methyl-1,3-oxazole-5-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
4-[2-(difluoromethoxy)benzoyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
9-[(4-chlorophenyl)methyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(5-cyanopyridin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-(1-{2-[2-(4-fluorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(prop-2-en-1-ylsulfanyl)propan-1-one
4-chloro-2-{[(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}phenol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
2-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-cyclopentyl-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(oxan-3-yl)acetamide
2-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-6-(trifluoromethyl)pyridine-3-carboxamide
4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]-1-(3-phenylpropyl)piperidin-4-ol
N-(3,5-dimethoxyphenyl)-3-{1-[2-(1H-imidazol-1-yl)acetyl]piperidin-3-yl}propanamide
5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
(1S,5R)-3-(2-methylquinolin-4-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[(2-chloro-4-fluorophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{2-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]phenyl}ethan-1-one
1-{6-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]pyridin-2-yl}ethan-1-ol
(2R)-2-cyclohexyl-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-hydroxyethan-1-one
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
(4aS,7aR)-1-(2-hydroxypyridine-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(2,3-difluorophenyl)methyl]-2-(5-ethyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-4-(1H-pyrazol-1-yl)benzamide
methyl 4-(4-{[2-(2-ethoxy-2-oxoethyl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
(1S,5R)-6-(4-fluoro-3-methylbenzoyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(furan-2-yl)ethyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-(furan-3-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
4-{[3-(2-aminoethyl)phenyl]methyl}-1-(2-methoxyphenyl)piperazin-2-one
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
4-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-{[3-(N-methylacetamido)pyrrolidin-1-yl]methyl}benzamide
(3S,4S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
methyl(propyl)({5-[2-(pyrrolidin-3-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclobutanecarbonylpyrrolidine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-2-(phenylamino)pyrimidine-5-carboxamide