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1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
3-chloro-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyridazine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-methyl-1,2-oxazol-5-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
1-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-tert-butyl-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-imidazole
4-{[4-(difluoromethoxy)phenyl]methyl}-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-({1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)-5-phenyl-2H-1,2,3,4-tetrazole
1-(2-{[(3R,4R)-4-hydroxy-1-(4-methoxybenzoyl)pyrrolidin-3-yl]amino}ethyl)imidazolidin-2-one
5-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenyl]-3-phenyl-1,2,4-oxadiazole
N,N-dimethyl-7-[(2-phenoxyethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2-(3-methoxyphenyl)piperidine
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
6-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
7-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-phenylacetamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-(2-phenylpyrrolidine-1-carbonyl)-2-(pyridin-4-yl)pyrimidine
3-[4-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-{[1-(2-fluorophenyl)cyclopropyl]methyl}piperidin-4-ol
N-cyclopropyl-2-[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-acetyl-6-methyl-3-[3-(2-methylpropyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-(2-amino-4-{[(5-methylpyrazin-2-yl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-hydroxyethan-1-one
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylpropane-1-sulfonamide
1-butyl-4-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperazin-2-one
2-methoxy-5-oxo-6-[3-(pyrrolidin-1-yl)propyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
6-(benzyloxy)-1-cyclohexyl-4-(5-methyl-1H-pyrazole-3-carbonyl)-1,4-diazepan-2-one
N,N-dimethyl-4-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)benzamide
(1R,2S)-2-propyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
1-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
8-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-amine
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[2-(benzylsulfanyl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
3-methyl-N-{3-[2-(4-methyl-1,4-diazepan-1-yl)acetamido]phenyl}benzamide
N-(2-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide
8-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]pyridine-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
7-(cyclopropylmethyl)-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(3-cyclopentylpropyl)-N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
(2S)-3-(1H-indol-3-yl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]propanoic acid
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-benzyl-N-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide