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N-[(5-{[2-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
N-methyl-N-(oxan-2-ylmethyl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3R,5S)-N-butyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-3-carboxamide
N,N-dimethyl-4-[4-({2-[2-(trifluoromethyl)phenyl]ethyl}amino)piperidin-1-yl]benzamide
2-{[4-(6-cyclopropylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
2-(2,4-dimethoxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
ethyl 4-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
methyl (1S,3S,3aR,6aS)-5-benzyl-3-(furan-3-yl)-1-(hydroxymethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5-(4-chlorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2,4-triazin-3-amine
(2R,3S,6R)-5-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)[1-(pyridin-3-yl)ethyl]amine
1-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidin-3-ol
ethyl 4-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylate
(1-{[methyl(pyridin-3-ylmethyl)amino]methyl}cyclopropyl)methanol
2-amino-3-ethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(4-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)acetamide
4-[(2,6-difluoro-3-methylphenyl)methyl]-1,4-oxazepan-5-one
N-(butan-2-yl)-5,7-dimethyl-N-(thiophen-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-(oxane-4-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
2,8-dimethyl-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
2-amino-4-[3-(4-chlorophenyl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-cyclohexyl-3-oxo-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
ethyl 5-({2-[5-(methylcarbamoyl)thiophen-2-yl]pyrrolidin-1-yl}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2-(1-propylpiperidin-4-yl)acetamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[2-({4-[(2,2-dimethyloxan-4-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
(1R,5S)-3-[(6-methoxy-2H-chromen-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,N-dimethyl-1H-pyrazole-4-carboxamide
N-(oxolan-3-yl)-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-4-(4-fluorophenyl)butane-1,4-dione
2-(4-hydroxyphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(2-methoxyphenyl)methyl]methylamine
4-(2,5-dihydro-1H-pyrrole-1-carbonyl)-2,7-dimethylquinoline
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-(hydroxymethyl)-1-(2-methylfuran-3-carbonyl)azepan-4-ol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
5-{1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4-methyl-1,2,3-thiadiazole
(4aS,8aR)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
5-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-ethylpyrimidine
2-(2-oxo-1,3-oxazolidin-3-yl)-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
3-(oxolan-3-yl)-5-(2-phenylphenyl)-1,2,4-oxadiazole
2-{4-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]butyl}pyridine
N-[2-(furan-2-yl)ethyl]-3-(1,4-oxazepane-4-sulfonyl)benzamide
N-(2-{7-propyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
(1R,9aR)-1-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-octahydro-1H-quinolizin-1-ol
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
(2S)-1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidine-2-carboxamide
1-cyclohexyl-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]piperidine-4-carboxamide