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N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]naphthalene-2-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
4-{3-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
4-(1H-1,3-benzodiazol-1-yl)-1-(propane-1-sulfonyl)piperidine-4-carboxylic acid
N-ethyl-N-[2-(4-fluorophenoxy)ethyl]-4-(hydroxymethyl)benzamide
N-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}methanesulfonamide
1-{1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperidin-4-yl}pyrrolidin-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxy-4-methylpentanamide
N-cycloheptyl-1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carboxamide
2-amino-6-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
2-[5-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
N-cyclopropyl-1-(2-{1-[2-(trifluoromethoxy)benzenesulfonyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
2-{methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}propane-1,3-diol
1-(2-methyl-1H-pyrrole-3-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
7-(2-hydroxyethyl)-2-[4-(1H-indol-3-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 3-(2,3-dimethylbenzoyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-2-fluorobenzamide
5-{4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}-1H-imidazol-2-amine
5-{[benzyl(methyl)amino]methyl}-N-[1-(methoxymethyl)cyclopropyl]-N-methyl-1,2-oxazole-3-carboxamide
7-(3-methoxy-2-methylbenzoyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
(2R,6R)-10-methoxy-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
7-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-3-methyl-3,4-dihydroquinazolin-4-one
5-methyl-N-{[3-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-benzyl-5-(cyclohex-3-en-1-ylmethyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(5-chloropyridin-2-yl)-4-(4,6-dimethylpyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(2,5-dimethylphenoxy)propyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-benzyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[4-(2,6-dimethoxypyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
3-chloro-5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-(2-ethoxypyridin-3-yl)acetic acid
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(6-methoxynaphthalen-2-yl)morpholine
3-(4-chloro-1H-pyrazol-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-{4-[2-(phenylsulfanyl)acetamido]-1H-pyrazol-1-yl}acetamide
1-{1-[2-(azepan-1-yl)-2-oxoethyl]piperidin-3-yl}-2-phenylethan-1-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[2-(2-ethylphenoxy)ethyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
4-(3-fluoro-4-methoxybenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-methyl-4-phenylthiophene-3-carboxamide
14-(2,3-dimethyl-1H-indol-7-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{4-[({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]piperidin-1-yl}ethan-1-ol
9-[(1-methyl-1H-imidazol-5-yl)methyl]-3-oxa-9-azaspiro[5.5]undecane
3-methyl-N-[1-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
4-[2-(2-chlorophenoxy)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1H-pyrazole-4-carboxamide