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3-(2-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethyl-1,3-oxazolidine-2,4-dione
1-[(4-fluorophenyl)methyl]-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-4-chloro-1,5-dimethyl-1H-pyrazole
N,N-diethyl-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidin-3-amine
3-[(2,4-difluorophenyl)methyl]-5-(4-methyl-1,3-oxazol-5-yl)-1,2,4-oxadiazole
9-benzoyl-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
(2S,4R)-4-{[(4-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-fluoro-N-({6-methyl-2-[methyl(1H-pyrazol-5-ylmethyl)amino]quinolin-3-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
(2R)-2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}-3-(3,4,5-trifluorophenyl)propanoic acid
2-methanesulfonyl-N-[2-methyl-1-(pyridin-2-yl)propyl]acetamide
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(pyridin-2-ylmethyl)-8-(pyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 5-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(4-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,5-dimethyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]isoquinoline
(4aS,8aR)-6-{[2-(carboxymethoxy)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
7-fluoro-4-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]quinazoline
1-[(5-methylfuran-2-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
5-(5-chloro-2-methylphenyl)-3-cyclopropyl-1H-1,2,4-triazole
(1R,5R)-3-(trimethylpyrimidin-4-yl)-3-azabicyclo[3.3.1]nonane
(3R,9aR)-3-methyl-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(piperidin-1-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(2,4-dimethylphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 4-(5-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-(furan-3-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
[5-(1-cyclopentyl-1H-imidazol-2-yl)-2-ethoxyphenyl]methanol
N-(2-methoxyethyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-cyclobutanecarbonyl-2-[(4-fluorophenyl)methyl]morpholine
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(1-methyl-1H-indol-5-yl)methyl]piperidin-3-yl]methanol
4-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridine
5-ethyl-2-methyl-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
(3S,4R)-4-phenyl-1-(quinoxaline-6-carbonyl)pyrrolidine-3-carboxylic acid
7-(2,2-dimethylpropyl)-2-[(4-fluoro-2-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
1-methyl-N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2,5-dimethylphenyl)methyl]-4-methylpiperidine
6-(4-fluorophenyl)-2-(3-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-{[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(methylsulfanyl)pyrimidine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-[(2-hydroxyethyl)(methyl)amino]-N-methylpyridine-3-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-phenylbenzamide
N-methyl-2-[methyl(pyridin-2-ylmethyl)amino]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-(1H-imidazol-5-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-(1H-pyrrol-1-yl)propan-1-one
3-[(4aR,7aS)-4-(morpholine-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid