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N2-(2-methoxyethyl)-N4-methyl-N4-[2-(pyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-cyclohexyl-N-(3,3-diphenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(phenylamino)-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}pyrimidine-5-carboxamide
4,5-dimethyl-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,3-dihydro-1,3-oxazol-2-one
N-(3-chloro-4-methoxyphenyl)-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
5-(2-methylpropyl)-1'-[(5-methylthiophen-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(1H-indol-3-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1-methylpiperidin-4-yl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]methanol
N-(1H-imidazol-2-ylmethyl)-N-methyl-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methyl-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
methyl 5-(dimethylsulfamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[3-(1,3-oxazol-5-yl)phenyl]urea
N-(1-cyanocyclohexyl)-3-(3,5-dimethylphenyl)propanamide
N,N-diethyl-3-(1-hydroxybutan-2-yl)-5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
(2S,4S)-4-amino-N-methyl-1-[1-(piperidin-1-yl)cyclohexanecarbonyl]pyrrolidine-2-carboxamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-4-(dimethylamino)butan-1-one
methyl 1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-4-carboxylate
2-(1,2,3,6-tetrahydropyridine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1H-imidazol-1-yl)ethyl]acetamide
4-(6-ethylpyrimidin-4-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]piperazine-1-carboxamide
3-methyl-6-(3-{1-[3-(pyridin-3-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyridazine
(3S)-4-{3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanoyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-(1-carbamoylcyclopentyl)-1-benzothiophene-5-carboxamide
1-(furan-2-ylmethyl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}piperidine-3-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1,2,5-tetramethyl-1H-pyrrole-3-carboxamide
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-3-methylthiophene-2-carboxamide
2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
1-cyclopentanecarbonyl-N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(1H-pyrazol-3-yl)pyridine-3-carboxamide
4-methyl-N-[1-(2-phenoxyacetyl)azepan-3-yl]piperazine-1-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-4-methyl-2-(methylamino)-1,3-thiazole-5-carboxamide
1,9-dimethyl-4-[2-(naphthalen-1-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)-1,3-oxazolidin-2-one
ethyl[(2-fluorophenyl)methyl](1H-imidazol-2-ylmethyl)amine
N-benzyl-N-methyl-3-[(3-propoxypiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
5-chloro-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thiophene-2-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(4,4,4-trifluorobutyl)pyrrolidine-2-carboxamide
1-[(1-acetylpiperidin-4-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
2,4-dimethyl-5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyrimidine
1-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-{furo[3,2-c]pyridin-4-yl}-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazine
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
2-[3,5-bis(trifluoromethyl)phenyl]-N,N-diethyl-4-hydroxypyrimidine-5-carboxamide
N-[(3S,4R)-1-(2-methylfuran-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
7-chloro-4-(1-methyl-1H-indole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3-methanesulfonamidophenyl)-3-[(2-methylphenyl)methoxy]azetidine-1-carboxamide
methyl 3-{7-chloro-2-[(furan-3-ylformamido)methyl]-2,3-dihydro-1-benzofuran-5-yl}benzoate