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3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(2,4-dimethoxyphenyl)ethyl]propanamide
1-(azepan-1-yl)-3-[2-methoxy-4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2-(4-fluorophenyl)-N-[2-(1H-imidazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(furan-2-yl)propan-1-one
4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
1-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
3-(3,5-dimethylphenyl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)propanamide
5-methyl-3-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-indole
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(prop-2-en-1-yl)acetamide
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,5-dimethoxybenzamide
5-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]benzonitrile
5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(5-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(thiophene-3-carbonyl)piperidine
N,N-dimethyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-(3-hydroxypropyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,2-dimethyl-1,3-thiazole-4-carboxamide
(1R,9aR)-1-({[(1S)-1-(3-methylpyridin-2-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
1-(furan-3-carbonyl)-4-[3-(1H-pyrazol-4-yl)benzoyl]-1,4-diazepane
2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]acetic acid
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-(prop-2-en-1-yl)benzamide
4-{4-[3-(2-methoxyphenoxy)azetidin-1-yl]pyridine-2-carbonyl}morpholine
3-tert-butyl-4-(4-methanesulfonylphenyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aR,7aS)-1-(3-methylbutanoyl)-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(1H-imidazol-1-yl)propanoyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethane-1,2-dione
1-tert-butyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrrole-3-carboxamide
1-(2-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyrimidin-4-yl)pyrrolidin-3-ol
(4S,4aS,8aS)-1-[(6-ethoxypyridin-3-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one
4-[(1-cycloheptylpiperidin-3-yl)sulfamoyl]benzoic acid
[(1-methyl-1H-pyrazol-4-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
5-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}-1-[(4-methylphenyl)methyl]azepan-2-one
ethyl 2-({3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl}amino)acetate
1-[1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-4-yl]piperidine-3-carboxylic acid
3-[(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]benzoic acid
8-(3-hydroxybenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl][(6-methoxypyridin-3-yl)methyl]methylamine
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-1,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1H-pyrazole-5-carboxamide
2-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethoxy}ethan-1-ol
5-ethyl-N-{1-oxaspiro[4.5]decan-3-yl}pyrimidin-2-amine
2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,3-dihydro-1,2-benzothiazol-3-one
8-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}-2,8-diazaspiro[4.5]decan-3-one
4-(pyridin-4-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrimidin-2-amine
(5-{1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
1-(2-hydroxy-3-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
ethyl 5-{[2-(1-benzyl-3-oxopiperazin-2-yl)acetamido]methyl}furan-2-carboxylate
2-{[2-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}-N-(2,4-dimethylphenyl)acetamide