Tips: Press Ctrl key to select multiple functional groups
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
5-methyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)pyrimidin-2-amine
dimethyl({2-[(oxolan-2-ylmethyl)({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]ethyl})amine
methyl 4-({[2-(5-oxo-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-yl)ethyl]amino}methyl)benzoate
ethyl (1R,9S)-5-amino-4-cyano-3-(3-ethyl-1H-pyrazol-5-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-12-carboxylate
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyridin-2-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
ethyl({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
(1S,6R)-3-methyl-9-[(1-methyl-1H-imidazol-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(thiophen-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[3-(4-{[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
(3S,4S)-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(4-fluorophenyl)piperidin-3-ol
N-[(3R,4R)-3-hydroxy-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl]pyridine-3-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
N-(2-tert-butyl-6-methylphenyl)-2-(trifluoromethyl)morpholine-4-carboxamide
8-ethoxy-5-{[3-(trifluoromethyl)phenyl]methyl}-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-(3-benzyl-1,2-oxazole-5-carbonyl)-3-(methoxymethyl)piperidine
1-ethyl-3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-(4-chloro-1H-indole-2-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(carbamoylmethyl)-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)piperidine-3-carboxamide
4-methoxy-6-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
2-(cyclohex-1-en-1-yl)-N-methylpyridine-3-carboxamide
2-(4-methoxyphenyl)-N-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
(2S,4R)-4-{[(2-chlorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-chloro-3-{[3-(4-ethylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-pyrazole
2-benzyl-9-(2-hydroxy-4-methylpentanoyl)-2,9-diazaspiro[5.5]undecan-3-one
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylmorpholine-4-sulfonamide
1-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
4-(cyclopropylmethyl)-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}butanamide
1-ethyl-6-oxo-N-[2-(quinolin-8-yloxy)ethyl]piperidine-3-carboxamide
[2,4,6-trimethyl-3-({[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}methyl)phenyl]methanol
2-[(4aR,7aS)-6,6-dioxo-4-(pent-2-yn-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
2-methyl-6-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-(3-hydroxypropyl)-1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-methyl-5-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(pyrimidin-2-yl)-4-[6-(thiophen-3-yl)pyridine-3-carbonyl]-1,4-diazepane
(2S)-N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-acetamidopropanamide
7-chloro-N-[(3R,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-4-hydroxyquinoline-3-carboxamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(morpholine-4-carbonyl)-1,4-diazepan-6-ol
(1S,6R)-9-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aR,7aS)-4-(1H-imidazol-4-ylmethyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methylacetamide
3-[1-(dimethylsulfamoyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]pent-4-en-1-one