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(1R,5S)-3-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3,8-diazabicyclo[3.2.1]octane
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(piperidin-1-yl)acetamide
N-(1-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
2-[(3-hydroxyazetidin-1-yl)methyl]-5,8-dimethylquinolin-4-ol
3,4-dimethyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-5-sulfamoylbenzamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2,7,8-trimethylquinoline-4-carboxamide
N-[(2-chlorophenyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(2-methoxyphenyl)-3-(1-{1-[3-(pyridin-4-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-ethoxy-6-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenol
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
4-[(3,5-dimethoxyphenyl)methyl]-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]quinoline-4-carboxylic acid
(3-{2-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
6-[3-(2-chlorophenyl)propanoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-{[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-N-methylfuran-2-carboxamide
{4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1,4-oxazepan-6-yl}methanol
N3-cyclooctyl-4-oxo-1-(pyridin-2-ylmethyl)-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(5-methoxyfuran-2-carbonyl)piperidine
1-(cyclobutylmethyl)-3-hydroxy-3-({[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
1-{1'-[2-(3-hydroxyphenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
({5-[1-(2,6-difluoro-4-methoxybenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-[(2-ethoxyphenyl)methyl]-3-(2-oxo-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)piperazin-2-one
(3aS,6aS)-2-(2-methoxyethyl)-5-[(4-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
8-cycloheptanecarbonyl-2-(propan-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N'-(3-fluorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}ethanediamide
3-(azepane-1-carbonyl)-1-(2-methylpropyl)-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridin-4-one
N-[(3-methoxyphenyl)methyl]-3-[1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)piperidin-3-yl]propanamide
5-propyl-2-(2,3,4-trimethoxyphenyl)pyrimidine
2-{1-[(4-ethoxyphenyl)methyl]-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl}ethan-1-ol
(2R,3S,6R)-5-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3S)-1-{4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanoyl}pyrrolidin-3-yl]acetamide
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
1-(2-methylpropyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-2-phenylmethanesulfonyl-1H-imidazole
(2S,4R)-4-amino-N,N-diethyl-1-[(4-methoxypiperidin-1-yl)sulfonyl]pyrrolidine-2-carboxamide
methyl[(2-methyl-1H-imidazol-4-yl)methyl]{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,5-dimethylfuran-3-carboxamide
2-{4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-1H-pyrazol-1-yl}ethan-1-ol
5-(3,4-difluorophenyl)-1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazole
4-chloro-3-({[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
ethyl 1-methanesulfonyl-4-(3-phenylpropyl)piperidine-4-carboxylate
6-{[(1S,2S)-2-hydroxycyclohexyl]amino}-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]thiophene-2-carboxamide
2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]pyridine-3-carboxylic acid
3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[2-(4-methylmorpholin-2-yl)ethyl]benzamide
3-(2-fluorophenoxymethyl)-N-(1-propyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
1-[(3R)-3-methylpiperazin-1-yl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-fluoro-3-(3-oxo-4-phenylpiperazine-1-carbonyl)benzene-1-sulfonamide