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N-({5-[(5-ethylpyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
4-chloro-5-{[3-(4-fluorophenoxy)azetidin-1-yl]methyl}-3-methyl-1H-pyrazole
5-(1H-imidazol-4-ylmethyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)acetamide
6-(dimethyl-1,2-oxazol-4-yl)pyridin-2-amine
4-(2-methoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N,N-dimethyl-2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethane-1-sulfonamide
N-ethyl-N-(oxan-4-ylmethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[2-(diethylamino)ethyl]-N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,3,4-thiadiazol-2-amine
3-[3-(5-methylfuran-2-yl)-5-[5-(propan-2-yl)-1,3-oxazol-4-yl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-(3-phenylpropyl)-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 3-[({[1-(phenoxymethyl)cyclopropyl]methyl}carbamoyl)amino]benzoate
6-fluoro-2-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}quinolin-4-ol
ethyl 3-[(3-chlorophenyl)methyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine-3-carboxylate
(4aS,7aR)-1-(4-hydroxybenzoyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
(4aR,8aR)-2-[2-(2-ethylphenoxy)ethyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[1-(methoxymethyl)cyclopropyl]-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)ethane-1-sulfonamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]cycloheptanamine
6-[1-(2-methoxyacetyl)piperidine-3-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(4-fluorophenyl)-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine
3-(1H-imidazol-1-ylmethyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(morpholin-3-yl)acetamide
1-{4-[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
4,5-dimethyl-6-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-(trifluoromethyl)pyrimidine
6-[(3-methoxyphenyl)methoxy]-4-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
(2S,4R)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-4-[(4-fluorophenyl)sulfanyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
4-{[3-(4-fluorophenoxy)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-(oxolan-3-ylmethyl)piperidine
1-cycloheptyl-N-[(2-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-{4-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(4-methylphenyl)propanamide
2-[1'-(furan-2-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
4-(3-chloro-4-methoxyphenyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[1-(4-{[2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]pyridine-3-carboxamide
4-methyl-1-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinolin-2-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methylpropyl)piperidine-4-carboxamide
3-(1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
3-(2-{[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]amino}ethyl)-1,3-oxazolidin-2-one
2-[methyl({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl})amino]ethan-1-ol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(oxan-4-ylmethyl)amino]methyl}piperidin-2-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(pent-4-enoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-carbamoylethyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide