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2-methyl-6-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-2,3-dihydropyridazin-3-one
2-[1-(6-aminopyridin-2-yl)-1H-pyrazol-4-yl]ethan-1-ol
3-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)pyridin-2-amine
N-methyl-2-(methylsulfanyl)-N-[(1-phenylpyrrolidin-3-yl)methyl]pyridine-3-carboxamide
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
6-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-2,3-dihydro-1,3-benzoxazol-2-one
(1R,9aR)-1-[(4,5-dichloro-1H-imidazol-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
4-(2,6-dimethylpyridin-3-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrimidin-2-amine
1-methyl-4-phenyl-5-(propan-2-yl)-1H-imidazole
methyl (2R,4S)-4-hydroxy-1-[2-(4-methoxy-3-methylphenyl)acetyl]piperidine-2-carboxylate
4,5-dimethyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
methyl 1-({8-methyl-2-[methyl(2-phenylethyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-4-carboxylate
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-oxopentanamide
1-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-2-phenoxyethan-1-one
1-methyl-5-[methyl(2-methylpropyl)amino]-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(cyclopentylamino)methyl]-N,N-diethylpyridin-2-amine
4-ethyl-3-{1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopentanecarboxamide
(1R,3S)-3-(2-aminoethoxy)-7-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-1-ol
8-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-ethyl-1H-pyrazole-5-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-4-(propan-2-yl)pyrimidin-2-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
(1S,5R)-3-(2,3-dihydro-1-benzofuran-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
2-(5-tert-butyl-1,3-benzoxazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-(3-phenylprop-2-ynoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-fluorophenyl)-N-(2-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(oxan-4-yl)acetamide
4-(2-methylpropyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
N-[2-(2-fluorophenoxy)ethyl]-2-(morpholin-2-yl)acetamide
3-(1-benzyl-5-oxopyrrolidin-3-yl)-1-[3-(2-methoxyethoxy)phenyl]urea
(1R,9aR)-N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-octahydro-1H-quinolizine-1-carboxamide
3,5-dimethyl-1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-3-yl]-1H-pyrazole
4-{2-[(E)-2-cyclohexylethenyl]pyridine-4-carbonyl}morpholine
(2R,3R,6R)-5-(dimethyl-1,3-thiazole-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
7-(1,2-oxazole-5-carbonyl)-2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
3-(2-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}ethyl)-4-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(aminomethyl)-N-[(1S)-1-cyclohexylethyl]-2-methylpyrimidin-4-amine
ethyl 1-(4-fluorophenyl)-5-(pyrrolidin-1-ylmethyl)-1H-pyrazole-4-carboxylate
N-(2-hydroxyethyl)-4-[(2-methylpyridin-3-yl)oxy]-N-propylpiperidine-4-carboxamide
2-chloro-4-({[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]carbamoyl}amino)-N-propylbenzamide
2-(4-{[2-(furan-2-yl)phenyl]methyl}morpholin-3-yl)-1-(pyrrolidin-1-yl)ethan-1-one
methyl 8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-(thian-4-yl)piperazine
(1R,9aR)-1-[({[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
(2S,4R)-1-[(5-methylfuran-2-yl)methyl]-4-[2-(methylsulfanyl)acetamido]-N-(propan-2-yl)pyrrolidine-2-carboxamide