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N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(3-methylthiophene-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-methyl-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]urea
4-(4-fluorobenzenesulfonyl)-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,4R)-1-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
methyl (2S,4R)-4-hydroxy-1-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)pyrrolidine-2-carboxylate
3-({[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}methyl)-1λ6-thiolane-1,1-dione
1-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)azetidine-3-carboxylic acid
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
1-methyl-6-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3-phenyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
6-methyl-N-(oxan-4-ylmethyl)-2-(piperidin-1-yl)pyrimidin-4-amine
4-{5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperazine-1-carbaldehyde
(3S,4S)-4-cyclopropyl-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
ethyl 1-(oxolane-2-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
7-methyl-4-(pyridin-4-yl)-6-(1H-1,2,4-triazole-5-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
(3S)-1-{7-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
2,5-dimethyl-N-[(4-sulfamoylphenyl)methyl]-1,3-thiazole-4-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
5-methoxy-1-methyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-indole-2-carboxamide
7-(3-methoxyphenyl)-2-(phenoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[1-(hydroxymethyl)-9-[2-(methylsulfanyl)acetyl]-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
1-(3-fluorophenyl)-5-(methoxymethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
1-[(3-fluorophenyl)methyl]-4-{[4-(2-hydroxyethoxy)phenyl]methyl}piperazin-2-one
3-(2-amino-4-methyl-6-{[2-(5-methylthiophen-2-yl)ethyl]amino}pyrimidin-5-yl)propanoic acid
6-methyl-2-{2-[(2-methyl-5-propylpyrimidin-4-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
5-{2-[(2-acetamidoethyl)amino]pyrimidin-4-yl}-2-ethoxybenzoic acid
3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
(4aS,7aR)-1-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(furan-3-ylmethyl)-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
1-{[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazol-2-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-[2-(4-methoxyphenyl)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
5-[({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
11-[(adamantan-2-ylmethyl)amino]-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
N-cyclopropyl-5-(3,5-difluoro-2-methoxyphenyl)thiophene-2-carboxamide
4-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
4-hydroxy-2-methyl-N-[1-(thian-4-yl)piperidin-4-yl]pyrimidine-5-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]benzamide
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-3-carboxamide
[(3aS,6aS)-2-(7-fluoro-2-methylquinoline-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-(1-cyclopentyl-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
methyl 1-{2-hydroxy-3-[4-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
8-[(5-ethylfuran-2-yl)methyl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(3-chlorophenyl)-1H-pyrazole-4-carboxylate
4-[(2,3-difluorophenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine