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4-{1-[(3-methylphenyl)methyl]-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl}pyridine
4-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
N-{1-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
1-[(3,4-dimethylphenyl)methyl]-4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]piperazin-2-one
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-[(1-cycloheptylpiperidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
3,3-dimethyl-1-{2-oxo-2-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}urea
4-ethyl-6-(4-{[(1-ethylpyrrolidin-2-yl)methyl]amino}piperidin-1-yl)-N,N-dimethylpyrimidin-2-amine
3-[1-(pyridin-3-yl)propan-2-yl]-5-(thiophen-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-N-[(1S,2R)-2-phenylcyclopropyl]piperidine-1-carboxamide
N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-methoxybenzamide
2-[2-({[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)piperidine-3-carboxamide
2-{2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
4-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}benzamide
[(4-ethyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-methyl-1-(2-oxo-2-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}ethyl)urea
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-ol
(2S)-2-amino-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzonitrile
(3S,4R)-4-(pyridin-3-yl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
N-[2-(azepan-1-yl)ethyl]-1-ethyl-6-methyl-2-oxo-N-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
4-[4-(4-fluorophenyl)-5-methyl-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
4-(4-chlorophenyl)-N-[2-(pyrazin-2-yl)ethyl]butanamide
N-[2-(4-methoxyphenyl)phenyl]-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide
4-(3-methylphenoxy)-1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
3-(4-fluorophenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
N-cyclohexyl-3-{[5-(4-methoxyphenyl)furan-2-yl]formamido}propanamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-[2-(thiomorpholin-4-ylmethyl)phenoxy]propanoic acid
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
(1S)-1-[1-(2-chlorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine
2-[(4-methoxyphenyl)methyl]-4-[4-(2-phenylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)ethan-1-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-[2-methoxy-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(1H-1,3-benzodiazole-5-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylic acid
4-methyl-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-1,2,3,6-tetrahydropyridine-1-carboxamide
ethyl 5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(3-fluorophenyl)-3-(furan-2-yl)-5-(2-methanesulfonylethyl)-1H-1,2,4-triazole
2-methyl-5-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
5-({3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-(pyridin-3-ylmethyl)piperidin-4-amine
4-chloro-3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
3-(ethylsulfanyl)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propan-1-one