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[(2S,4R)-4-(dimethylamino)-1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]methanol
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazole
[(dimethyl-1,2-oxazol-4-yl)methyl](1-phenoxypropan-2-yl)amine
4-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidine-3-carboxamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
(3R,4S)-4-[(1-benzothiophen-3-ylmethyl)(methyl)amino]oxolan-3-ol
ethyl 4-benzyl-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate
N-[(3S,4R)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
({4-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine
(2E)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-methylbut-2-enamide
1-(4-fluorophenyl)-N-(thiolan-3-yl)cyclopropane-1-carboxamide
3-{4-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenyl}prop-2-yn-1-ol
7-(1,3-benzothiazol-2-yl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-acetyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-2-carboxamide
N-ethyl-5-{[methyl(quinolin-5-ylmethyl)amino]methyl}pyrimidin-2-amine
2-[({5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methyl)sulfanyl]pyrimidine
4-(1H-imidazol-1-yl)-1-(2-methylbenzenesulfonyl)piperidine-4-carboxylic acid
7-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2H-1,3-benzodioxole-5-carboxamide
[5-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
2-methoxy-N-[1-(thian-4-yl)piperidin-4-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
5-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-N'-(2-ethoxyphenyl)propanediamide
2-methyl-5-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]pyrazine
2-(5-methyl-1H-pyrazol-1-yl)-1-{9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
3,4,7-trimethyl-2-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-indole
8-{[2-(4-fluorophenyl)ethyl]carbamoyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-6-(2,3,6-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(thian-4-yl)piperazine
4-hydroxy-2-{[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}quinoline-6-carboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[2-(pyridin-4-yl)ethyl]propanamide
(2S)-2-{4-[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}-3-methylbutanamide
N-benzyl-N-methyl-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-amine
ethyl 2-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-2-yl}acetate
N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-1-yl)benzamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-5-ylmethyl)benzamide
8-methyl-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3,4-dihydroquinazolin-4-one
2-methyl-3-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,8-naphthyridine
6-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carbonitrile
2-(dimethylamino)-6-(2-methylphenyl)-N-(thiophen-2-ylmethyl)pyridine-3-carboxamide
1-(2-chlorophenyl)-2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethan-1-ol
1,3-dimethyl-2,6-dioxo-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(2-{[2-(1H-indol-3-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-cycloheptylpiperidine-1-carboxamide
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide