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(2S,4R)-4-amino-N,N-diethyl-1-methanesulfonylpyrrolidine-2-carboxamide
1-(3-methylpyridin-2-yl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazine
(3aR,6aR)-N-(2-methoxyethyl)-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
3-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,6-dimethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-({1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}methyl)furan-2-carboxamide
N-(4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenyl)acetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
4-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)morpholine
2-cyclopropyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrimidine
9-(2,6-dimethoxypyrimidine-4-carbonyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(2-phenoxyethyl)propanamide
(1R,3s,6r,8S)-4-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
5-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
5-ethyl-2,3-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-{1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}pyridine
4-[1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
3-(3-methoxyphenyl)-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(2-cyclohexylethyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
2-cyclohexyl-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-cyclopentanecarbonyl-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
3-(2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)imidazolidine-2,4-dione
4-(1H-imidazol-1-yl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-4-carboxylic acid
5-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-methyl-1H-indol-1-yl)propanamide
[(2S)-1-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidin-2-yl]methanol
(3S)-N-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-3-(3-methoxyphenyl)piperidine-1-carboxamide
N'-cyclopentyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)butanediamide
3-(4-methylpiperazin-1-yl)-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridazine
(4aR,7aS)-1-{2-[methyl(thiophen-2-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({[(5-methylfuran-2-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
3-(2-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-4-methyl-4H-1,2,4-triazole
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-fluoro-4-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridine
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
5-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
(3aR,6aR)-2-methanesulfonyl-N-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
4-(piperidin-1-yl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]butan-1-one
4-{5-[2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]phenol
2-(4-fluoro-3-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
3-methyl-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
1-ethyl-3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide