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1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-[(2-fluorophenyl)methoxy]azetidine
(1S,5R)-6-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
1-[3-(4-{[(1-ethylpyrrolidin-2-yl)methyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-(pyridine-2-carbonyl)piperidin-4-amine
6-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}-N-(2H-1,3-benzodioxol-5-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2-methylphenyl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
9-(2-amino-6-methoxypyrimidin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 5-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-(2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)-1H-1,2,4-triazole
1-(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-(3-chloro-2-methylphenyl)-3-(2-methoxybenzoyl)piperidine-1-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-methyl-6-oxo-N-[(3R,5S)-1-(pent-2-yn-1-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1,6-dihydropyridazine-3-carboxamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)-4-(2-methoxyethyl)piperazine
1-(propan-2-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
3-fluoro-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
(3S,9aR)-3-(cyclohexylmethyl)-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[2-chloro-5-(trifluoromethoxy)phenyl]-N-cyclopropylfuran-2-carboxamide
N-(3,4-difluorophenyl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-amine
2-{[5-(1,3-dimethyl-1H-pyrazol-5-yl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[3-(methylsulfanyl)propyl]benzamide
ethyl 4-[2-(2,6-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]piperidine-1-carboxylate
(benzylsulfamoyl)(methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
N-ethyl-3-(2-fluorophenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
2-ethoxy-5-[2-(pyridin-3-yl)pyrimidin-4-yl]benzoic acid
methyl 5-(2,6-dimethoxypyrimidine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[(3,5-dimethoxyphenyl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-N-methylpyrrolidine-3-carboxamide
5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-3-propyl-1H-pyrazole
2-(dimethylamino)-2-(4-fluorophenyl)-N-(1H-indol-5-ylmethyl)acetamide
N3-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N3-methylpiperidine-1,3-dicarboxamide
5-benzyl-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3-chloro-4-fluorophenyl)-3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}propanamide
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(piperidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
9-(5,6-dimethylpyrimidin-4-yl)-6-oxa-9-azaspiro[4.5]decane
N-(propan-2-yl)-5-(1H-pyrazol-4-yl)thiophene-2-carboxamide
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-[2-(trifluoromethyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[1'-(5-amino-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-(1,4-dithiepan-6-yl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-(2-methanesulfonylethyl)-3-(phenoxymethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-[(3R,4S)-4-(morpholin-4-yl)-1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]propanoic acid
4-{2-[(3-chloro-4-fluorophenyl)carbamoyl]ethyl}-N-(2-methoxyethyl)piperidine-1-carboxamide
3-{1-[1-(4-fluorophenyl)cyclopropyl]-N-(pyridin-3-ylmethyl)formamido}propanoic acid
N-[2-(4-fluorophenyl)-1-{1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
N-[3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}amino)phenyl]cyclopentanecarboxamide