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(3S,4R)-1-(3-methanesulfonamidopropanoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[2-(1H-imidazol-1-yl)ethyl]-3-({[3-(2-methylphenyl)phenyl]methyl}amino)-5-(pyrrolidine-1-sulfonyl)benzamide
1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-3-phenylpiperidine
1-(4-methoxyphenyl)-4-[1-(oxane-4-carbonyl)piperidin-3-yl]piperazine
1-(4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)butan-1-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-ol
N-ethyl-5-(4-methoxyphenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]furan-2-carboxamide
7-(2-methoxyethyl)-2-(naphthalen-1-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(1H-imidazol-4-yl)-1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazole
3-[2-(3-fluorophenyl)ethyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
6-cyclopropyl-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]pyrimidin-4-amine
4-{[(1R)-1-carbamoylethyl]sulfamoyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-methyl-1-{[3-(2-phenylazetidine-1-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
(3S,9aR)-3-[(benzyloxy)methyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclohexyl-1-cyclopropyl-6-oxopiperidine-3-carboxamide
N-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)-2-methylpropanamide
N,N-dimethyl-2-{[(oxan-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-N,N-dimethyl-4-oxobutanamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-[(6-methoxypyridin-3-yl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
N-[2-(furan-2-ylmethoxy)phenyl]-2-methylpyrrolidine-1-carboxamide
2-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
(2E)-3-(3-fluorophenyl)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
3-(furan-2-yl)-1-[4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
N3-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-1,3-dicarboxamide
3-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
3-hydroxy-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
2-(benzyloxy)-1-[6-hydroxy-4-(3-hydroxypropyl)-1,4-diazepan-1-yl]ethan-1-one
2-{2-[1-(azepane-1-sulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
5-[2-(propan-2-yl)-1H-imidazol-1-yl]quinoline
2-methoxy-N-(2-methyl-3-{[(propan-2-yl)(2,2,2-trifluoroethyl)carbamoyl]amino}phenyl)acetamide
[(3R,4R)-1-[(2,6-difluorophenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]pyridine-3-sulfonamide
5-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}amino)-2-methoxy-N,N-dimethylbenzamide
2-methyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzofuran-5-carboxamide
1'-(3-methyl-1H-pyrazole-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-(3-acetylphenyl)-3-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}urea
2-(cyclopropylmethyl)-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(2-phenylethyl)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-N-[(1s,4s)-4-aminocyclohexyl]piperidine-3-carboxamide
N-{2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
N-({1-[2-(morpholin-4-yl)-2-oxoethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)thiophene-2-carboxamide
3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-(2-oxopyrrolidin-1-yl)-N-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]propanamide
N-(1-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)benzamide
(1S,3R)-3-amino-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}cyclopentane-1-carboxamide
2-(methylsulfanyl)-4-(2,4,6-trimethylphenyl)pyrimidine
N-[(3S,4R)-4-(4-methylphenyl)-1-(thiophene-3-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide