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3-[(cyclohexylamino)methyl]-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-[(3-methyl-1H-indol-2-yl)methyl]pyridazin-3-amine
1-ethyl-2-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
(3aS,6aS)-2-(oxan-4-yl)-5-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
2-{benzyl[1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethan-1-ol
4-(3-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]oxy}benzoyl)morpholine
N-[2-(dimethylsulfamoyl)ethyl]-2-methyl-1,3-benzothiazole-5-carboxamide
N-(4-{1-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
2-methyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]phenol
1-[1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
7-(1H-indol-5-ylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
6-ethyl-4-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)-2H-chromen-2-one
N-(3-fluoro-5-methylphenyl)-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
2-[4-(morpholin-4-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
1-[3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-(3-acetylphenyl)-6-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(oxolan-2-ylmethyl)-9-(pyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(dimethyl-1,2-oxazol-4-yl)acetamide
2-(dimethylamino)-1-{3-[2-(pyridin-3-yl)pyridin-4-yl]pyrrolidin-1-yl}ethan-1-one
4-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
9-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-[(5-ethyl-1-benzofuran-3-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-(2-chlorophenyl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methylfuran-2-carboxamide
N-[(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)methyl]thiophene-2-sulfonamide
1-[2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidine-3-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
2-ethyl-9-[2-(2-hydroxyethoxy)ethyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-(1-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-methylpropan-2-yl)morpholine
5-(4-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenyl)-1,3,4-thiadiazol-2-amine
N,7-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
(4aR,7aS)-1-benzyl-4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1,3-thiazol-2-yl)piperidin-3-yl]methanol
1-{1'-[3-(5-methylfuran-2-yl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(pyrrolidin-1-yl)ethan-1-one
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3,3-diphenylpiperidine
1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(5S,9aS,9bS)-5-(furan-2-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-ethyl-4,6-dimethyl-2-oxo-N-[(2,3,4-trifluorophenyl)methyl]-1,2-dihydropyridine-3-carboxamide
2-methyl-6-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
4-{3-cyclopropyl-5-[2-(1H-1,2,4-triazol-3-yl)phenyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,5S,6R)-3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-[(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-{3-[3-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one