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2-{4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperazin-1-yl}pyrazine
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
[(2,5-dimethylphenyl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-{1-[1-(3-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-2-methylpropyl}acetamide
3-(2,6-dimethoxypyridin-3-yl)-1-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)urea
1-[(2S,4R)-1-{[3-(2-methylphenyl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
4-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(4-methoxyphenyl)piperazin-2-one
1-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-3-methylbutan-1-one
1-cyclohexyl-4-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperazine
5-(3-methoxyphenoxymethyl)-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
4-(furan-3-yl)-N,6-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
7-[3-(2-hydroxyphenyl)propanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1,4-dimethyl-9-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]-1,4,9-triazaspiro[5.5]undecane
2-[(3,5-difluorophenyl)methyl]-8-[2-(dimethylamino)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(1H-imidazol-2-yl)benzamide
1-{1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
(4aS,7aR)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(4-chlorophenoxy)ethyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-chlorophenyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]morpholine
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
3-[(3R,4S)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carboxamide
1-[2-(4-fluoro-2-methylphenyl)acetyl]-N-(4-fluorophenyl)piperazine-2-carboxamide
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
1-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pentane-1,2-dione
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)propylamine
2-methoxy-2-phenyl-1-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetamide
1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
3-cyclopentaneamido-4-methyl-N-[2-(pyridin-3-yloxy)propyl]benzamide
N-(1-{2-[(4S,4aS,8aR)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-phenoxyacetamide
4-[(5-ethylpyridin-2-yl)methyl]-2-[(3-fluorophenyl)methyl]morpholine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-N-ethylacetamide
3-{1-[2-(morpholin-4-yl)ethyl]piperidin-3-yl}benzoic acid
3-(methoxymethyl)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}benzamide
1-(3-fluoro-4-methoxybenzoyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
3-[1-(7-chloroquinoxalin-2-yl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-3-(4-methylpiperazine-1-carbonyl)-2-propyl-1,4-dihydropyridin-4-one
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-1-(2-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-{[2-(3-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(4-methoxy-3,5-dimethylphenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
{4-[(3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
1-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-pyrazole-3-carboxamide
1-cyclopentyl-4-{2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}piperazin-2-one
1-{2-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
6-[(3-methylpiperidin-1-yl)methyl]-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide