Varenicline-d4 Tartrate

• Catalog No.: V098492
• M. F.: C17H19N3O6
• M. W.: 361.34926

SYNONYMS

• IUPAC name: (13,13,15,15-^2H₄)-5,8,14-triazatetracyclo[10.3.1.0^2,^1^1.0^4,^9]hexadeca-2,4,6,8,10-pentaene; 2,3-dihydroxybutanedioic acid
• IUPAC Traditional name: (.+-.)-tartaric acid; (13,13,15,15-^2H₄)-5,8,14-triazatetracyclo[10.3.1.0^2,^1^1.0^4,^9]hexadeca-2,4,6,8,10-pentaene
• Synonyms: CP 526555-18-d4; 7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine (2R,3R)-2,3- Dihydroxybutanedioate-d4; Champix-d4

DETAILS

Description (English)

Labelled nicotinic α4β2 acetylcholine receptor partial agonist. Aid in smoking cessation.

REFERENCES

• Benowitz, N., et al.: Clin. Pharmacol. Ther., 44, 23 (1988)
• Cohen, C., et al.: J. Pharmacol. Exp. Ther., 306, 407 (1988)
• Tapper, A., et al.: Science, 306, 1029 (1988)
• Coe, J., et al.: J. Med. Chem., 48, 3474 (1988)
• Obach, R., et al.: Drug Metab. Disp