Triptorelin Acetate

• Catalog No.: T815800
• CAS Number: 140194-24-7
• M. F.: C66H86N18O15
• M. W.: 1371.50064
• Storage: Hygroscopic, -20°C Freezer, Under inert atmosphere

SYNONYMS

• IUPAC name: (2S)-N-[(2S)-5-carbamimidamido-1-[(2S)-2-[(carbamoylmethyl)carbamoyl]pyrrolidin-1-yl]-1-oxopentan-2-yl]-2-[(2R)-2-[(2S)-2-[(2S)-3-hydroxy-2-[(2S)-2-[(2S)-3-(1H-imidazol-5-yl)-2-{[(2S)-5-oxopyrrolidin-2-yl]formamido}propanamido]-3-(1H-indol-3-yl)propanamido]propanamido]-3-(4-hydroxyphenyl)propanamido]-3-(1H-indol-3-yl)propanamido]-4-methylpentanamide; acetic acid
• IUPAC Traditional name: (2S)-N-[(2S)-5-carbamimidamido-1-[(2S)-2-(carbamoylmethylcarbamoyl)pyrrolidin-1-yl]-1-oxopentan-2-yl]-2-[(2R)-2-[(2S)-2-[(2S)-3-hydroxy-2-[(2S)-2-[(2S)-3-(3H-imidazol-4-yl)-2-{[(2S)-5-oxopyrrolidin-2-yl]formamido}propanamido]-3-(1H-indol-3-yl)propanamido]propanamido]-3-(4-hydroxyphenyl)propanamido]-3-(1H-indol-3-yl)propanamido]-4-methylpentanamide; acetic acid
• Synonyms: BIM 21003C; 6-D-Tryptophan Luteinizing Hormone-Releasing Factor (Swine) Acetate; 6-D-Tryptophan Luteinizing Hormone-Releasing Factor (Pig) Acetate; Decapeptyl-Depot; OvuGel

DATABASE IDS

• CAS Number: 140194-24-7

PROPERTIES

• Apperance: White Solid
• Melting Point: >222°C (dec.)
• Solubility: Methanol
• Solubility: Water
• Storage Condition: Hygroscopic, -20°C Freezer, Under inert atmosphere

DETAILS

Description (English)

Synthetic peptide agonist analog of LH-RH. Triptoreline is a potent agonist of LH-releasing hormone, currently used in the treatment of prostatic cancer where therapy may be required over months or years. Antineoplastic (hormonal). Used in the treatment o

REFERENCES

• Sanders, L., et al.: Eur. J. Drug Metab. Pharmacokinet., 15, 95 (1990)
• Chiba, M., et al.: Biomaterials, 18, 893 (1990)
• Blanco, D., et al.: Eur. J. Pharm. Biopharm., 45, 285 (1990)
• Sinha, V., et al.: J. Control. Rel., 90, 261 (1990)