Δ4-Tibolone-13C,d3

• Catalog No.: T437507
• M. F.: C21H28O2
• M. W.: 313.43847484
• Storage: -20°C Freezer

SYNONYMS

• IUPAC name: (1R,2R,9S,10R,11S,14R,15S)-14-ethynyl-14-hydroxy-9-(^1^3C,^2H₃)methyl-15-methyltetracyclo[8.7.0.0^2,^7.0^1^1,^1^5]heptadec-6-en-5-one
• IUPAC Traditional name: (1R,2R,9S,10R,11S,14R,15S)-14-ethynyl-14-hydroxy-9-(^1^3C,^2H₃)methyl-15-methyltetracyclo[8.7.0.0^2,^7.0^1^1,^1^5]heptadec-6-en-5-one
• Synonyms: 7α-Methylnorethindrone-13C,d3; NSC 142228-13C,d3; 17α-Ethynyl-17-hydroxy-7α-(methyl-13C,d3)-4-estren-3-one; (7α,17α)-17-Hydroxy-7-(methyl-13C,d3)-19-norpregn-4-en-20-yn-3-one; Org-OM 38-13C,d3

PROPERTIES

• Apperance: White Solid
• Melting Point: 188-190°C`
• Solubility: Chloroform
• Storage Condition: -20°C Freezer

DETAILS

Description (English)

A labelled metabolite of Tibolone. A synthetic steroid with weak estrogenic, androgenic and progestogenic activity. A pharamceutical used in the treatment of menopausal syndrome.

REFERENCES

• Clarkson, T., et al.: J. Clin. Endocrinol. Metab., 86, 5396 (2001)
• Landgren, M., et al.: Maturitas, 50, 222 (2001)
• Wang, M., et al.: Steroids, 71, 343 (2001)
• Verheul, H., et al.: Drug Metab. Dispos., 35, 1105 (2001)