Tianeptine

• Catalog No.: T436800
• CAS Number: 72797-41-2
• M. F.: C21H25ClN2O4S
• M. W.: 436.9522
• Storage: Refrigerator, Under Inert Atmosphere

SYNONYMS

• IUPAC name: 7-({6-chloro-10-methyl-9,9-dioxo-9λ^6-thia-10-azatricyclo[9.4.0.0^3,^8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}amino)heptanoic acid
• IUPAC Traditional name: tianeptine
• Synonyms: (+/-)-7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide; Coaxil; 7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide

DATABASE IDS

• CAS Number: 72797-41-2

PROPERTIES

• Apperance: White Solid
• Melting Point: 129-131°C
• Solubility: DMSO
• Solubility: Methanol
• Solubility: Water
• Storage Condition: Refrigerator, Under Inert Atmosphere

DETAILS

Description (English)

Tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Antidepressant.

REFERENCES

• Malen, C., et al.: Experientia, 28, 811 (1972)
• Safa, A., et al.: J. Biol. Chem., 262, 7884 (1972)
• Ford, J.M., et al.: Pharmacol. Rev., 42, 155, (1972)
• Pierre, A., et a.: Cancer Res., 51, 2312 (1972)