Thiocolchicoside-d3

• Catalog No.: T344387
• M. F.: C27H33NO10S
• M. W.: 563.61662

SYNONYMS

• IUPAC name: N-[(10S)-3,4-dimethoxy-14-(methylsulfanyl)-13-oxo-5-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}tricyclo[9.5.0.0^2,^7]hexadeca-1(16),2(7),3,5,11,14-hexaen-10-yl](^2H₃)acetamide
• IUPAC Traditional name: N-[(10S)-3,4-dimethoxy-14-(methylsulfanyl)-13-oxo-5-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}tricyclo[9.5.0.0^2,^7]hexadeca-1(16),2(7),3,5,11,14-hexaen-10-yl](^2H₃)acetamide
• Synonyms: Coltrax-d3; Miorel-d3; Coltramyl-d3; (S)-N-[3-(β-D-Glucopyranosyloxy)-5,6,7,9-tetrahydro-1,2-dimethoxy-10-(methylthio)-9-oxobenzo[a]heptalen-7-yl]acetamide-d3; N-[(7S)-3-(β-D-Glucopyranosyloxy)-5,6,7,9-tetrahydro-1,2-dimethoxy-10-(methylthio)-9-oxobenzo[a]heptalen-7-yl]acetamide-d3; Miotens-d3; Muscoril-d3; NSC 147755-d3

DETAILS

Description (English)

A labelled GABA receptor antagonist which is prescribed as a muscle relaxant having analgesic effects.

REFERENCES

• Gelmi, M., et al.: J. Med. Chem., 50, 2245 (2007)
• Mascia, M., et al.: Eur. J. Pharmacol., 558, 37 (2007)
• Gohil, V., et al.: Nat. Biotechnol., 28, 249 (2007)