Thiocolchicoside

• Catalog No.: T344385
• CAS Number: 602-41-5
• M. F.: C27H33NO10S
• M. W.: 563.61662
• Storage: Refrigerator

SYNONYMS

• IUPAC name: N-[(10S)-3,4-dimethoxy-14-(methylsulfanyl)-13-oxo-5-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}tricyclo[9.5.0.0^2,^7]hexadeca-1(16),2(7),3,5,11,14-hexaen-10-yl]acetamide
• IUPAC Traditional name: thiocolchicoside
• Synonyms: Coltramyl; NSC 147755; Miorel; Muscoril; Coltrax; N-[(7S)-3-(β-D-Glucopyranosyloxy)-5,6,7,9-tetrahydro-1,2-dimethoxy-10-(methylthio)-9-oxobenzo[a]heptalen-7-yl]acetamide; (S)-N-[3-(β-D-Glucopyranosyloxy)-5,6,7,9-tetrahydro-1,2-dimethoxy-10-(methylthio)-9-oxobenzo[a]heptalen-7-yl]acetamide; Miotens

DATABASE IDS

• CAS Number: 602-41-5

PROPERTIES

• Apperance: Yellow solid
• Melting Point: 190-198°C
• Solubility: Water
• Storage Condition: Refrigerator

DETAILS

Description (English)

A GABA receptor antagonist which is prescribed as a muscle relaxant having analgesic effects.

REFERENCES

• Gelmi, M., et al.: J. Med. Chem., 50, 2245 (2007)
• Mascia, M., et al.: Eur. J. Pharmacol., 558, 37 (2007)
• Gohil, V., et al.: Nat. Biotechnol., 28, 249 (2007)