Tapentadol O-β-D-Glucuronide

• Catalog No.: T007210
• CAS Number: 1300037-86-8
• M. F.: C20H31NO7
• M. W.: 397.46264
• Storage: Hygroscopic, -20°C Freezer, Under Inert Atmosphere

SYNONYMS

• IUPAC name: (2S,3S,4S,5R,6S)-6-{3-[(2R,3R)-1-(dimethylamino)-2-methylpentan-3-yl]phenoxy}-3,4,5-trihydroxyoxane-2-carboxylic acid
• IUPAC Traditional name: (2S,3S,4S,5R,6S)-6-{3-[(2R,3R)-1-(dimethylamino)-2-methylpentan-3-yl]phenoxy}-3,4,5-trihydroxyoxane-2-carboxylic acid
• Synonyms: 3-[(1R,2R)-3-(Dimethylamino)-1-ethyl-2-methylpropyl]phenyl β-D-Glucopyranosiduronic Acid

DATABASE IDS

• CAS Number: 1300037-86-8

PROPERTIES

• Apperance: White to Off-White Solid
• Melting Point: >170°C (dec.)
• Solubility: Methanol
• Solubility: Water
• Storage Condition: Hygroscopic, -20°C Freezer, Under Inert Atmosphere

DETAILS

Description (English)

A metabolite of Tapentadol (T007200).

REFERENCES

• Terlinden, R., et al.: Eur. J. Drug Metab. Pharmacokinet., 32, 163 (2007)
• Tzschentke, T., et al.: J. Pharmacol. Exp. Ther., 323, 256 (2007)
• Wade, W., et al.: Clin. Ther., 31, 2804 (2007)