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Linagliptin

Catalog No. L465900 Name Toronto Research Chemicals
CAS Number 668270-12-0 Website http://www.trc-canada.com
M. F. C25H28N8O2 Telephone +1 (416) 665-9696
M. W. 472.54222 Fax +1 (416) 665-4439
Purity Email info@trc-canada.com
Storage Refrigerator Chembase ID: 172303

SYNONYMS

IUPAC name
8-[(3R)-3-aminopiperidin-1-yl]-7-(but-2-yn-1-yl)-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]-2,3,6,7-tetrahydro-1H-purine-2,6-dione
IUPAC Traditional name
linagliptin
Synonyms
BI 1356BS
8-[(3R)-3-Amino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-1H-purine-2,6-dione
BI 1356
ONDERO
8-[(3R)-3-Amino-1-piperidinyl]-7-(2-butynyl)-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-1H-purine-2,6-dione

DATABASE IDS

CAS Number 668270-12-0

PROPERTIES

Certificate of Analysis Download
Apperance Yellowish Orange Solid
Melting Point 190-196°C (dec.)
Solubility DMSO
Solubility Methanol
MSDS Link Download
Storage Condition Refrigerator

DETAILS

Description (English)
A novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.

REFERENCES

  • Prabavathy, N. et al.: Int. J. Pharm. Bio. Sci., 2, 438 (2011)
  • Deacon, C.F.: Diab. Obes. Metab., 13, 7 (2011)